SCHEMBL6081383

SCHEMBL6081383

O=c1n(-c2ccc(NCCCNCC3CC3)cc2)ccn1-c1ccc(OC2CCCC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
TSHR P16473 1/20 0.39
HRH3 Q9Y5N1 7/20 0.37
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
CTSL P07711 2/20 0.35
CTSS P25774 2/20 0.35
CTSK P43235 2/20 0.35
ACACB O00763 2/20 0.35
ACACA Q13085 1/20 0.35
P2RX3 P56373 2/20 0.35
FFAR4 Q5NUL3 2/20 0.35
NAMPT P43490 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080987 0.88 ALDH1A1 (0.43) ALDH1A1TSHRHRH3CTSLCTSS
SCHEMBL6081705 0.83 HRH3 (0.39) ALDH1A1TSHRHRH3CTSLCTSS
SCHEMBL6081381 0.81 HRH3 (0.38) ALDH1A1TSHRHRH3ACACBACACA
SCHEMBL6082261 0.80 CYP19A1 (0.42) ALDH1A1TSHRKDM4E
SCHEMBL1728613 0.75 HRH3 (0.46) ALDH1A1TSHRHRH3ACACB
SCHEMBL6081179 0.73 HRH3 (0.41) ALDH1A1HRH3KDM4EACACB
SCHEMBL6081508 0.72 KDM4E (0.50) ALDH1A1TSHRHRH3KDM4E
SCHEMBL1728644 0.72 HRH3 (0.42) ALDH1A1TSHRHRH3KDM4EACACB
SCHEMBL6081904 0.72 HRH3 (0.42) ALDH1A1TSHRHRH3KDM4EACACB
SCHEMBL1727601 0.71 KDM4E (0.52) ALDH1A1HRH3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7141561-B2 Substituted diaryl heterocycles, process for their preparation and their use as medicaments SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-11-28 US disclosed
US-20040132752-A1 Substituted diaryl heterocycles, process for their preparation and their use as medicaments AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-07-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040132752-A1 Substituted diaryl heterocycles, process for their preparation and their use as medicaments GPR119, GLP1R, SLC5A2 ALDH1A1 1096/4885TSHR 919/4885HRH3 1710/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.