SCHEMBL6081969

SCHEMBL6081969

Cc1ccccc1COc1ccc(-n2ccn(-c3ccc(OCCN(C)C)cc3)c2=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 6/20 0.57
KCNH2 Q12809 4/20 0.47
MAPK14 Q16539 1/20 0.46
MAOB P27338 1/20 0.45
MAPT P10636 1/20 0.44
LTA4H P09960 2/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
FGFR1 P11362 1/20 0.41
SRC P12931 1/20 0.41
FFAR1 O14842 1/20 0.41
TNKS O95271 1/20 0.41
ACHE P22303 1/20 0.40
S1PR1 P21453 1/20 0.39
S1PR5 Q9H228 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1728493 0.84 MCHR1 (0.78) MCHR1KCNH2LTA4HFGFR1SRC
SCHEMBL1728515 0.84 MCHR1 (0.52) MCHR1KCNH2MAPK14LTA4HCYP1A2
SCHEMBL6082151 0.82 MCHR1 (0.60) MCHR1KCNH2MAPK14LTA4HCYP1A2
SCHEMBL1728669 0.82 LTA4H (0.68) MCHR1KCNH2MAPK14LTA4HCYP1A2
SCHEMBL1728477 0.81 MCHR1 (0.56) MCHR1KCNH2MAPK14MAPTCYP1A2
SCHEMBL1728621 0.81 MCHR1 (0.63) MCHR1KCNH2MAPK14MAOBMAPT
SCHEMBL6080985 0.80 MCHR1 (0.54) MCHR1MAPK14LTA4HCYP1A2CYP2D6
SCHEMBL6081903 0.80 MCHR1 (0.54) MCHR1KCNH2MAPK14LTA4HCYP1A2
SCHEMBL6081522 0.80 ALDH1A1 (0.55) MCHR1KCNH2MAPK14MAPTLTA4H
SCHEMBL1728658 0.80 LTA4H (0.70) MCHR1KCNH2LTA4HCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7141561-B2 Substituted diaryl heterocycles, process for their preparation and their use as medicaments SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-11-28 US disclosed