SCHEMBL6087563

SCHEMBL6087563

Nc1cnn(-c2cccnn2)c1N

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.41
CYP1A2 P05177 1/20 0.41
SCN9A Q15858 1/20 0.36
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
GOT1 P17174 1/20 0.33
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33
OPRM1 P35372 1/20 0.31
OPRL1 P41146 1/20 0.31
SMPD3 Q9NY59 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL26127628 0.78 CYP17A1 (0.36) CYP17A1CYP1A2SCN9A
SCHEMBL27700574 0.78 RIPK2 (0.47) NPC1RAB9ATP53HPGD
SCHEMBL11338402 0.78 RIPK2 (0.57) CYP17A1CYP1A2NPC1RAB9ATP53
SCHEMBL3252316 0.76 RAB9A (0.52) CYP17A1CYP1A2NPC1RAB9ATP53
Hydrochloric Acid SCHEMBL5415490 0.75 RAB9A (0.51) CYP17A1CYP1A2NPC1RAB9ATP53
Hydrochloric Acid SCHEMBL6087752 0.75 RAB9A (0.51) CYP17A1CYP1A2NPC1RAB9ATP53
SCHEMBL14688311 0.71 CYP17A1 (0.35) CYP17A1CYP1A2SCN9AGOT1
SCHEMBL10561233 0.71 NPC1 (0.72) CYP1A2NPC1RAB9ATP53HPGD
SCHEMBL6087110 0.70 HTR3E (0.41) CYP1A2NPC1RAB9AHPGD
SCHEMBL6087909 0.70 MAPT (0.45) CYP17A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7056354-B2 Compounds derived from diaminopyrazole substituted by a heteroaromatic radical and their use in oxidation dyeing of keratinous fibers L'OREAL (FR) 2006-06-06 US claimed
US-20040255397-A1 Compounds derived from diaminopyrazole substituted by a heteroaromatic radical and their use in oxidation dyeing of keratimous fibers L'OREAL (FR) 2004-12-23 US claimed
EP-1412348-A1 COMPOUNDS DERIVED FROM DIAMINOPYRAZOLE SUBSTITUTED BY A HETEROAROMATIC RADICAL AND THEIR USE IN OXIDATION DYEING OF KERATINOUS FIBRES L'OREAL (FR) 2004-04-28 EP claimed
WO-2003008405-A1 COMPOUNDS DERIVED FROM DIAMINOPYRAZOLE SUBSTITUTED BY A HETEROAROMATIC RADICAL AND THEIR USE IN OXIDATION DYEING OF KERATINOUS FIBRES L'OREAL (FR) 2003-01-30 WO claimed
US-7056354-B2 Compounds derived from diaminopyrazole substituted by a heteroaromatic radical and their use in oxidation dyeing of keratinous fibers L'OREAL (FR) 2006-06-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040255397-A1 Compounds derived from diaminopyrazole substituted by a heteroaromatic radical and their use in oxidation dyeing of keratimous fibers KRT18, AOC1, XRCC5 CYP17A1 1146/4885CYP1A2 250/4885SCN9A 3765/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.