SCHEMBL6089628

SCHEMBL6089628

COC(c1cn(Cc2ccc3ccccc3n2)cn1)c1cccc(C)c1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYSLTR1 Q9Y271 9/20 0.37
GPBAR1 Q8TDU6 3/20 0.37
SIRT2 Q8IXJ6 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
CYSLTR2 Q9NS75 7/20 0.35
CYP1A2 P05177 1/20 0.35
ALOX5 P09917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6092667 0.81 PTGDR2 (0.37) CYSLTR1GPBAR1PTGDR2CYSLTR2CYP1A2
SCHEMBL6089639 0.77 CYSLTR1 (0.41) CYSLTR1GPBAR1SIRT2PTGDR2CYSLTR2
SCHEMBL6089338 0.69 CYP1A2 (0.37) CYSLTR1GPBAR1SIRT2CYSLTR2CYP1A2
SCHEMBL6090578 0.67 CYSLTR1 (0.58) CYSLTR1GPBAR1CYSLTR2CYP1A2ALOX5
SCHEMBL6089645 0.66 CYSLTR1 (0.39) CYSLTR1GPBAR1CYSLTR2CYP1A2ALOX5
SCHEMBL3875985 0.65 MLKL (0.48)
SCHEMBL6089838 0.65 CYSLTR1 (0.46) CYSLTR1GPBAR1CYSLTR2CYP1A2ALOX5
SCHEMBL6092671 0.65 CYSLTR1 (0.39) CYSLTR1GPBAR1PTGDR2CYSLTR2CYP1A2
SCHEMBL6088426 0.65 CYSLTR1 (0.46) CYSLTR1GPBAR1CYSLTR2CYP1A2
SCHEMBL5725146 0.64 CYSLTR1 (0.67) CYSLTR1GPBAR1CYSLTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7005440-B1 Therapeutic uses of tri-aryl acid derivatives AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2006-02-28 US disclosed