SCHEMBL6089771

SCHEMBL6089771

N#CCOc1c(Cl)cc(Cl)cc1COc1cccc(O)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 4/20 0.43
NR4A1 P22736 1/20 0.43
NR4A3 Q92570 1/20 0.43
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HPD P32754 1/20 0.39
APP P05067 1/20 0.39
CHRNB4 P30926 2/20 0.36
CHRNA3 P32297 2/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
POLB P06746 1/20 0.36
ALOX15 P16050 1/20 0.36
HTT P42858 1/20 0.36
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6090588 0.88 NR4A2 (0.39) NR4A2NR4A1NR4A3NPC1RAB9A
SCHEMBL6088014 0.78 CYSLTR1 (0.51)
SCHEMBL28107564 0.78 CHRNB2 (0.50) APPCHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL5725097 0.77 CHRNB2 (0.40) NR4A2NR4A1NR4A3NPC1RAB9A
SCHEMBL6088015 0.75 CYSLTR1 (0.42)
SCHEMBL6088663 0.75 POLB (0.43) POLBALOX15HTT
SCHEMBL11276165 0.74 NR4A2 (0.68) NR4A2NR4A1NR4A3NPC1RAB9A
SCHEMBL6089396 0.72 POLB (0.40) POLBALOX15HTT
SCHEMBL7398355 0.68 GRM5 (0.50) NR4A2HTTMAOB
SCHEMBL15607572 0.67 FFAR1 (0.52) NR4A2NPC1RAB9AAPPCHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7005440-B1 Therapeutic uses of tri-aryl acid derivatives AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2006-02-28 US disclosed
EP-1177176-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS Aventis Pharma Deutschland GmbH (DE) 2002-02-06 EP disclosed
WO-2000064876-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-11-02 WO disclosed