SCHEMBL609186

SCHEMBL609186

CC(C)OC(=O)N1CCC(OCc2noc(-c3ccc(N4CC[C@H](c5cc(F)ccc5F)[C@@H](NC(=O)C(C)(C)C)C4)nc3)n2)CC1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 6/20 0.35
HRH3 Q9Y5N1 5/20 0.34
RET P07949 5/20 0.33
CETP P11597 1/20 0.32
PPARG P37231 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32
DGAT1 O75907 1/20 0.32
NTRK1 P04629 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10058409 0.89 DPP4 (0.39) GPR119HRH3
Hydrochloric Acid SCHEMBL611275 0.88 DPP4 (0.39) GPR119HRH3
Hydrochloric Acid SCHEMBL611820 0.88 DPP4 (0.39) GPR119HRH3
SCHEMBL612843 0.83 GPR119 (0.35) GPR119CETPNTRK1
SCHEMBL10058402 0.79 MCHR1 (0.36) GPR119CETPPPARGPPARDPPARA
SCHEMBL609509 0.78 GPR119 (0.39) GPR119HRH3
SCHEMBL13186827 0.78 GPR119 (0.39) GPR119HRH3
SCHEMBL10058410 0.78 GPR119 (0.43) GPR119HRH3
Hydrochloric Acid SCHEMBL612832 0.77 GPR119 (0.42) GPR119HRH3
SCHEMBL13186640 0.77 GPR119 (0.43) GPR119HRH3RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120040953-A1 Compounds for the Treatment of Metabolic Disorders PROSIDION LIMITED (GB) 2012-02-16 US disclosed
EP-2406256-A1 COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS Prosidion Limited (GB) 2012-01-18 EP disclosed
WO-2010103335-A1 COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS PROSIDION LIMITED (GB) 2010-09-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120040953-A1 Compounds for the Treatment of Metabolic Disorders GPR119, GPR132, FFAR2 GPR119 1/4885HRH3 793/4885RET 1439/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.