SCHEMBL6092800

SCHEMBL6092800

NCCNC(=O)C1CCN(Cc2ccc(Cl)cc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
ACKR3 P25106 2/20 0.53
MAPT P10636 1/20 0.53
TSHR P16473 1/20 0.53
HTT P42858 1/20 0.53
HRH3 Q9Y5N1 1/20 0.53
CYP2D6 P10635 1/20 0.52
CHRM4 P08173 1/20 0.52
TP53 P04637 1/20 0.50
POLB P06746 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2262431 0.88 CHRM4 (0.65) ALDH1A1TSHRCYP2D6CHRM4POLB
SCHEMBL7486412 0.81 ALDH1A1 (0.58) ALDH1A1ACKR3POLB
SCHEMBL5368002 0.79 GAA (0.69) ALDH1A1MAPTHTTHRH3
SCHEMBL30924045 0.78 ACKR3 (0.62) ACKR3HTT
SCHEMBL2073212 0.77 DRD2 (0.60) ALDH1A1MAPTHTTHRH3
SCHEMBL14124454 0.76 ACHE (0.63) ALDH1A1HTT
SCHEMBL21820693 0.76 TEAD1 (0.58) ALDH1A1MAPTHTT
SCHEMBL19554726 0.76 KDM4E (0.72) ALDH1A1TSHRCHRM4
SCHEMBL6705571 0.75 ALDH1A1 (0.61) ALDH1A1MAPTTSHRHTTCYP2D6
SCHEMBL6093929 0.75 DRD2 (0.54) ALDH1A1MAPTHTTCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7125895-B1 Cyclic amine derivatives and their uses BRISTOL-MYERS SQUIBB PHARMA RESEARCH LABS, INC. (US) 2006-10-24 US disclosed
EP-1181278-B1 CYCLIC AMINE DERIVATIVES AND THEIR USES BRISTOL MYERS SQUIBB PHARMA RE (US) 2004-09-29 EP disclosed