SCHEMBL609296

SCHEMBL609296

CC(C)OC(=O)N1CCC(OCc2nc(-c3cnc(Cl)nc3)no2)CC1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 10/20 0.55
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ACACB O00763 1/20 0.39
ACACA Q13085 1/20 0.39
LMNA P02545 2/20 0.38
FAAH O00519 2/20 0.38
KCNH2 Q12809 1/20 0.37
CYP11B2 P19099 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPK1 P28482 1/20 0.37
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL612271 0.91 GPR119 (0.56) GPR119ACACBACACALMNAFAAH
SCHEMBL609466 0.90 GPR119 (0.55) GPR119CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL610359 0.90 GPR119 (0.54) GPR119ACACBACACALMNAFAAH
SCHEMBL386190 0.85 GPR119 (0.76) GPR119CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL10058389 0.83 GPR119 (0.39) GPR119FAAH
SCHEMBL610385 0.82 GPR119 (0.51) GPR119ACACBACACAFAAH
SCHEMBL4424816 0.81 GPR119 (0.58) GPR119SMN1; SMN2ALDH1A1
SCHEMBL10058416 0.77 GPR119 (0.44) GPR119CYP2C9ACACBACACALMNA
SCHEMBL609646 0.77 GPR119 (0.73) GPR119CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL10058411 0.77 GPR119 (0.44) GPR119CYP2C9HTTSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102395584-A Compounds for the treatment of metabolic disorders PROSIDION LTD 2012-03-28 CN disclosed
US-20120040953-A1 Compounds for the Treatment of Metabolic Disorders PROSIDION LIMITED (GB) 2012-02-16 US disclosed
US-20120040953-A1 Compounds for the Treatment of Metabolic Disorders PROSIDION LIMITED (GB) 2012-02-16 US disclosed
US-20120040953-A1 Compounds for the Treatment of Metabolic Disorders PROSIDION LIMITED (GB) 2012-02-16 US disclosed
EP-2406256-A1 COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS Prosidion Limited (GB) 2012-01-18 EP disclosed
WO-2010103335-A1 COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS PROSIDION LIMITED (GB) 2010-09-16 WO disclosed
WO-2010103335-A1 COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS PROSIDION LIMITED (GB) 2010-09-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120040953-A1 Compounds for the Treatment of Metabolic Disorders GPR119, GPR132, FFAR2 GPR119 1/4885CYP1A2 1452/4885CYP2D6 1922/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.