SCHEMBL6092970

SCHEMBL6092970

COC(=O)c1ccc(C(=O)Cc2cc(-c3cccs3)ccc2OCCN2CCCCC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
ESR1 P03372 7/20 0.47
ESR2 Q92731 7/20 0.47
MCHR1 Q99705 6/20 0.46
MEN1 O00255 1/20 0.45
GAA P10253 1/20 0.45
KMT2A Q03164 1/20 0.45
KCNH2 Q12809 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
ATM Q13315 2/20 0.41
NPC1 O15118 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
NR4A2 P43354 1/20 0.40
GLA P06280 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PPARG P37231 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6091297 0.90 KCNH2 (0.47) KDM4EESR1ESR2MCHR1KCNH2
SCHEMBL6092086 0.86 SMN1; SMN2 (0.46) MEN1GAAKMT2ANPC1RAB9A
SCHEMBL6092548 0.82 KDM4E (0.50) KDM4EMEN1KMT2AATMNPC1
SCHEMBL6110229 0.81 LTA4H (0.42) KDM4EMEN1KMT2AATMNPC1
SCHEMBL6092689 0.78 MAPT (0.45) KDM4EMEN1KMT2AATMNPC1
SCHEMBL6094350 0.77 TNFRSF1A (0.45) KDM4EMEN1GAAKMT2ANPC1
SCHEMBL6092917 0.76 SMN1; SMN2 (0.43) MEN1GAAKMT2ANPC1RAB9A
SCHEMBL6094179 0.74 HRH3 (0.56) KDM4EESR1ESR2MCHR1KCNH2
SCHEMBL6092780 0.73 TNFRSF1A (0.50) KDM4EMEN1KMT2A
SCHEMBL6091940 0.73 TNFRSF1A (0.52) KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060063828-A1 1,2-Bis-(substituted-phenyl)-2-propen-1-ones and pharmaceutical compositions thereof ATHEROGENICS, INC. 2006-03-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060063828-A1 1,2-Bis-(substituted-phenyl)-2-propen-1-ones and pharmaceutical compositions thereof ABCB11, CEL, CYP46A1 KDM4E 1931/4885ESR1 3626/4885ESR2 2668/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.