SCHEMBL6094700

SCHEMBL6094700

O=C1C=C(O)C(=O)C(c2c[nH]c3cc(Br)ccc23)=C1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.45
CCNE2 O96020 1/20 0.43
CDK4 P11802 1/20 0.43
CCND1 P24385 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
CYP2A6 P11509 1/20 0.41
ADRA1A P35348 4/20 0.41
ADRA1B P35368 4/20 0.41
CLK1 P49759 3/20 0.40
CDK5 Q00535 2/20 0.40
CDK5R1 Q15078 2/20 0.40
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
PRKACA P17612 1/20 0.40
PRKACG P22612 1/20 0.40
PRKACB P22694 1/20 0.40
CSNK1A1 P48729 1/20 0.40
CSNK1D P48730 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6096806 0.90 EGFR (0.44) CLK1CDK5CDK5R1CCNB2CDK1
SCHEMBL6096484 0.84 IDH1 (0.41) CDK4CCND1GSK3BIDO1PTPN1
SCHEMBL6095097 0.84 TDO2 (0.46) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL6094665 0.84 NR4A2 (0.41) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL6097125 0.81 PRKCB (0.54) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL6095741 0.78 TSHR (0.40) PTPN1
SCHEMBL6099085 0.76 KDM4E (0.44) IDO1PTPN1
SCHEMBL6096702 0.76 IGF1R (0.44) CAMK2DIDO1
SCHEMBL6096745 0.76 F7 (0.44) CAMK2DIDO1PTPN1
SCHEMBL6096063 0.75 RET (0.40) CDK4CCND1CDK2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7057052-B2 Heterocyclic quinones as pharmaceutical agents DUKE UNIVERSITY (US) 2006-06-06 US disclosed
WO-2004050014-A2 SETEROCYCLIC QUINONES AS PHARMACEUTICAL AGENTS DUKE UNIVERSITY (US) 2004-06-17 WO disclosed
US-20040063774-A1 Heterocyclic quinones as pharmaceutical agents DUKE UNIVERSITY 2004-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063774-A1 Heterocyclic quinones as pharmaceutical agents NQO1, RECQL, SDHA IMPDH2 218/4885CCNE2 91/4885CDK4 106/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.