SCHEMBL6094728

SCHEMBL6094728

Cn1c(N2CCN(CCOCCO)CC2)nc(C(=O)NCc2ccc(F)cc2)c(O)c1=O

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNE1 P15382 1/20 0.45
CCR1 P32246 1/20 0.45
KCNQ1 P51787 1/20 0.45
HTR1A P08908 6/20 0.44
HTR7 P34969 6/20 0.44
KCNH2 Q12809 1/20 0.44
CYP2C9 P11712 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
DRD2 P14416 4/20 0.42
HTR6 P50406 4/20 0.42
LIPG Q9Y5X9 2/20 0.41
CALCA P06881 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6093565 0.91 KCNE1 (0.49) KCNE1CCR1KCNQ1KCNH2CYP2C9
SCHEMBL6094040 0.89 MMP13 (0.41) KCNE1CCR1KCNQ1HTR1AHTR7
SCHEMBL6093724 0.87 KCNE1 (0.49) KCNE1CCR1KCNQ1KCNH2CYP2C9
SCHEMBL6094737 0.84 CYP2C9 (0.56) KCNE1CCR1KCNQ1KCNH2CYP2C9
SCHEMBL6094550 0.84 KCNH2 (0.54) KCNE1CCR1KCNQ1KCNH2CYP2C9
SCHEMBL12776746 0.83 CYP2C9 (0.55) KCNE1CCR1KCNQ1KCNH2CYP2C9
SCHEMBL6094768 0.83 KCNE1 (0.49) KCNE1CCR1KCNQ1KCNH2CYP2C9
SCHEMBL6094863 0.82 MEN1 (0.52) KCNE1CCR1KCNQ1HTR7KCNH2
SCHEMBL6093745 0.82 KCNE1 (0.52) KCNE1CCR1KCNQ1KCNH2CYP2C9
SCHEMBL6094821 0.82 KCNE1 (0.50) KCNE1CCR1KCNQ1KCNH2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7135467-B2 Pyrimidine carboxamides; 5-hydroxy-2-(2-(1,1-Dioxo-6-[1,2]thiazinan-2-yl)-6-oxo-1,6-dihydropyrimidine-4-carboxamides; AIDS; AIDS related complex BRISTOL-MYERS SQUIBB COMPANY (US) 2006-11-14 US disclosed
US-20040204498-A1 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2004-10-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040204498-A1 HIV integrase inhibitors IMPDH1, TYMP, REV1 KCNE1 3935/4885CCR1 660/4885KCNQ1 4594/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.