Mephenoxalone

Mephenoxalone

SCHEMBL6098064

COc1ccccc1OCC1CNC(=O)O1.COc1ccccc1OCC1CNC(=O)O1.S

nearest known ligand 0.75

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.75
SYK P43405 8/20 0.58
ADRA2C P18825 1/20 0.54
LMNA P02545 2/20 0.53
MAOA P21397 1/20 0.53
SLC6A2 P23975 1/20 0.53
IRAK4 Q9NWZ3 2/20 0.53
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
MAPT P10636 1/20 0.47
USP2 O75604 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mephenoxalone SCHEMBL4621926 0.99 PKM (0.77) PKMSYKADRA2CLMNAMAOA
Mephenoxalone SCHEMBL935967 0.99 PKM (0.77) PKMSYKADRA2CLMNAMAOA
Mephenoxalone SCHEMBL5392 0.99 PKM (0.77) PKMSYKADRA2CLMNAMAOA
Mephenoxalone SCHEMBL1969509 0.97 PKM (0.75) PKMSYKADRA2CLMNAMAOA
Mephenoxalone SCHEMBL1061349 0.97 PKM (0.75) PKMSYKADRA2CLMNAMAOA
Mephenoxalone SCHEMBL22472152 0.97 PKM (0.75) PKMSYKADRA2CLMNAMAOA
Mephenoxalone SCHEMBL2175454 0.97 PKM (0.75) PKMSYKADRA2CLMNAMAOA
Mephenoxalone SCHEMBL7117835 0.97 PKM (0.75) PKMSYKADRA2CLMNAMAOA
Mephenoxalone SCHEMBL7938104 0.97 PKM (0.75) PKMSYKADRA2CLMNAMAOA
Mephenoxalone SCHEMBL6492968 0.96 PKM (0.73) PKMSYKADRA2CLMNAMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7002020-B1 Oxazolidinone combinatorial libraries, compositions and methods of preparation PHARMACIA & UPJOHN COMPANY (US) 2006-02-21 US disclosed
US-20050004174-A1 Antibacterial agents GORDEEV MIKHAIL F (US) 2005-01-06 US disclosed
US-6562844-B2 Attaching an olefin to a solid support; oxidizing the olefin to provide an epoxide functionality; opening the epoxide with an amine to form an amino alcohol; cyclizing the amino alcohol using a phosgene equivalent PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed
US-6531470-B1 Antimicrobial compounds PHARMACIA & UPJOHN COMPANY 2003-03-11 US disclosed
US-20020183371-A1 Oxazolidinone combinatorial libraries, compositions and methods of preparation GORDEEV MIKHAIL F (US) 2002-12-05 US disclosed
US-6239152-B1 Oxazolidinone combinatorial libraries, compositions and methods of preparation PHARMACIA & UPJOHN COMPANY 2001-05-29 US disclosed
EP-1049682-A1 OXAZOLIDINONE COMBINATORIAL LIBRARIES, COMPOSITIONS AND METHODS OF PREPARATION Versicor, Inc. (US) 2000-11-08 EP disclosed
WO-1999037630-A1 OXAZOLIDINONE COMBINATORIAL LIBRARIES, COMPOSITIONS AND METHODS OF PREPARATION VERSICOR, INC. (US) 1999-07-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020183371-A1 Oxazolidinone combinatorial libraries, compositions and methods of preparation PAICS, CDK4, OXA1L PKM 147/4885SYK 56/4885ADRA2C 4178/4885
US-20050004174-A1 Antibacterial agents PAICS, OXA1L, PNKP PKM 600/4885SYK 171/4885ADRA2C 4737/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.