Triaziquone

Triaziquone

SCHEMBL610295

NCCN.O=C1C=C(N2CC2)C(=O)C(N2CC2)=C1N1CC1

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3PDE3APDE3BPDE4APDE4BPDE4CPDE4D

The experimentally established mechanism targets of Triaziquone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNMT1 P26358 1/20 0.42
MAPT P10636 2/20 0.40
HTT P42858 2/20 0.40
TP53 P04637 1/20 0.40
STAT3 P40763 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
APAF1 O14727 2/20 0.35
TDP2 O95551 2/20 0.35
NSD2 O96028 2/20 0.35
HKDC1 Q2TB90 2/20 0.35
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
GALK1 P51570 1/20 0.33
BLM P54132 1/20 0.33
ATM Q13315 1/20 0.33
NOD2 Q9HC29 1/20 0.33
ATG4B Q9Y4P1 1/20 0.33
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triaziquone SCHEMBL2160619 0.98 DNMT1 (0.41) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL10379983 0.98 DNMT1 (0.41) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL11416072 0.96 DNMT1 (0.40) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL600168 0.93 DNMT1 (0.40) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL6830995 0.91 DNMT1 (0.39) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL3700755 0.91 DNMT1 (0.39) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL1961248 0.91 DNMT1 (0.39) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL33439 0.91 HTT (0.42) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL11428634 0.91 DNMT1 (0.41) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL5800741 0.91 DNMT1 (0.41) DNMT1MAPTHTTTP53STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 332 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250154662-A1 THERMAL ATOMIC LAYER ETCHING PROCESSES ASM IP HOLDING B.V. (NL) 2025-05-15 US claimed
US-12252590-B2 Acetoacetylated and (meth)acrylated resin compositions and thermosets and foams therefrom NDSU RESEARCH FOUNDATION (US) 2025-03-18 US claimed
US-12227738-B2 Method of single-stranded RNA purification SARTORIUS BIA SEPARATIONS D.O.O. (SI) 2025-02-18 US claimed
CN-114773307-B Non-isocyanate polyurethane monomer and thermosetting non-isocyanate shape memory polyurethane, and preparation and recycling methods thereof 中国科学院兰州化学物理研究所 2024-01-26 CN claimed
US-20220290005-A1 COATINGS WITH TUNABLE AMINE DENSITY Cowper Sciences Inc. 2022-09-15 US claimed
CN-114773307-A Non-isocyanate-based polyurethane monomer and thermosetting non-isocyanate-based shape memory polyurethane, and preparation and recycling methods thereof 中国科学院兰州化学物理研究所 2022-07-22 CN claimed
CN-113527313-B Preparation method and application of water-soluble supermolecule organic cage-shaped compound for detecting pyridinium substances in water 浙江浙能技术研究院有限公司 2022-07-12 CN claimed
CN-109906489-B Flexible electrode and method for producing a flexible electrode 高丽大学校产学协力团 2022-02-25 CN claimed
US-11168284-B2 Laundry builders and surfactants derived from bio-based hydroxyacids and epoxides BATTELLE MEMORIAL INSTITUTE (US) 2021-11-09 US claimed
CN-113527313-A Preparation method and application of water-soluble supermolecule organic cage-shaped compound for detecting pyridinium substances in water 浙江浙能技术研究院有限公司 2021-10-22 CN claimed
US-20040132993-A1 Antiviral and antimicrobial guanidine or biguanidine derivatives SHETTY B VITHAL (US) 2004-07-08 US claimed
US-20020042495-A1 Polyamide ligand-containing polymeric resins and methods of using the same for removing, separating and/or concentrating desired metal ions from solutions BRUENING RONALD L (US) 2002-04-11 US claimed
JP-2001507724-A 2001-06-12 JP claimed
EP-0411774-B2 Improvements to multifilament apparel yarns of nylon DU PONT (US) 2000-06-21 EP claimed
EP-0979266-A2 NOVEL WATER SOLUBLE METAL WORKING FLUIDS Solutia Inc. (US) 2000-02-16 EP claimed
WO-1998008919-A2 NOVEL WATER SOLUBLE METAL WORKING FLUIDS SOLUTIA INC. (US) 1998-03-05 WO claimed
US-5202182-A Used in hosiery E. I. DU PONT DE NEMOURS AND COMPANY (US) 1993-04-13 US claimed
US-5137666-A Nylon 66 modified with nylon 6 monomer or 2-methyl-pentamethylenediamine; hosiery E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-08-11 US claimed
EP-0411774-A1 Improvements to multifilament apparel yarns of nylon E.I. DU PONT DE NEMOURS AND COMPANY (US) 1991-02-06 EP claimed
US-4847315-A SOLUTION POLYMERIZATION OF TRIS/2-AMINOETHYL/AMINE, DECYANDIAMIDE, FORMALDEHYDE AND DICARBOXYLIC ACID AND/OR EPTICHLOROHYDRIN; ALKYL KETENE DIMER EMULSIONS W. R. GRACE AB (SE) 1989-07-11 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040132993-A1 Antiviral and antimicrobial guanidine or biguanidine derivatives GMPS, GDA, GANC DNMT1 746/4885MAPT 3246/4885HTT 2457/4885
US-20220290005-A1 COATINGS WITH TUNABLE AMINE DENSITY CHRM1, C5, CHRM2 DNMT1 71/4885MAPT 1384/4885HTT 2097/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.