SCHEMBL6119280

SCHEMBL6119280

CS(=O)(=O)Nc1cc2oc(-c3ccc(C(F)(F)F)cc3)c(C(=O)O)c2cc1C1CC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 4/20 0.40
CYP2C9 P11712 4/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2C19 P33261 3/20 0.40
KCNH2 Q12809 2/20 0.40
ANO1 Q5XXA6 2/20 0.39
KIF11 P52732 2/20 0.38
FPR1 P21462 3/20 0.38
FPR2 P25090 3/20 0.38
SLC22A12 Q96S37 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
KDM1A O60341 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6119825 0.91 CYP2C9 (0.49) CYP2C9CYP3A4CYP2C19KCNH2KIF11
SCHEMBL2295568 0.89 CYP2C9 (0.48) CYP2C9CYP3A4CYP2C19KCNH2ANO1
SCHEMBL2296799 0.87 CYP2C9 (0.43) CYP2C9CYP3A4CYP2C19KCNH2ANO1
SCHEMBL6119722 0.85 CYP2C9 (0.45) CYP2C9CYP3A4CYP2C19KCNH2ANO1
SCHEMBL2302690 0.84 CYP2C9 (0.45) CYP2C9CYP3A4CYP2C19KCNH2ANO1
SCHEMBL6120266 0.83 CYP2C9 (0.41) TRPV1CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2298467 0.81 CYP2C9 (0.47) CYP2C9CYP3A4CYP2C19KCNH2ANO1
SCHEMBL6120327 0.80 CYP2C9 (0.46) CYP2C9CYP3A4CYP2C19KCNH2ANO1
SCHEMBL2298808 0.80 CYP2C9 (0.59) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2298218 0.80 CYP2C9 (0.48) CYP2C9CYP3A4CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012067663-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-05-24 WO disclosed