SCHEMBL6120945

SCHEMBL6120945

CNC(=O)c1c(-c2ccc(F)cc2)nn2cc(NS(=O)(=O)CCc3ccccc3)c(OC)cc12

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.39
KMT2A Q03164 3/20 0.38
MAPT P10636 3/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 2/20 0.38
NTSR1 P30989 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
APLNR P35414 3/20 0.37
BRAF P15056 2/20 0.37
EDNRB P24530 1/20 0.37
EDNRA P25101 1/20 0.37
CYP17A1 P05093 1/20 0.37
PTGS2 P35354 1/20 0.35
TP53 P04637 1/20 0.35
MDM2 Q00987 1/20 0.35
HPGD P15428 1/20 0.35
PI4KB Q9UBF8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6120998 0.93 ACLY (0.43) ACLYKMT2AMAPTKDM4EALDH1A1
SCHEMBL2994042 0.86 BRAF (0.44) BRAF
SCHEMBL17332238 0.85 BRD4 (0.38) KMT2AMAPTALDH1A1LMNABRAF
SCHEMBL6121072 0.84 MAPT (0.36) MAPTALDH1A1BRAF
SCHEMBL3000942 0.81 BRAF (0.43) BRAF
SCHEMBL2994199 0.80 BRAF (0.46) BRAF
SCHEMBL6120949 0.80 L3MBTL1 (0.43) KMT2AMAPTKDM4EALDH1A1LMNA
SCHEMBL17332257 0.79 BRAF (0.37) LMNABRAFHPGD
SCHEMBL2987982 0.78 BRAF (0.44) MAPTBRAFTP53
SCHEMBL2998731 0.78 BRAF (0.46) BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012067664-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-05-24 WO disclosed