SCHEMBL6125232

SCHEMBL6125232

Bc1ccc(NC)c(C#N)c1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
CDC42BPA Q5VT25 1/20 0.37
CDC42BPB Q9Y5S2 1/20 0.37
ABCC9 O60706 1/20 0.31
ABCC8 Q09428 1/20 0.31
KCNJ11 Q14654 1/20 0.31
KCNJ8 Q15842 1/20 0.31
TSHR P16473 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17194144 0.78 ALDH1A1 (0.42) ROCK2ROCK1CDC42BPACDC42BPBTSHR
SCHEMBL28381748 0.78 LOXL2 (0.41) ROCK2ROCK1CDC42BPACDC42BPB
SCHEMBL9230994 0.76 LRRK2 (0.40) ROCK2ROCK1CDC42BPACDC42BPB
SCHEMBL20375313 0.76 SRC (0.39) ROCK2ROCK1CDC42BPACDC42BPBTSHR
SCHEMBL11829926 0.76 KDM4E (0.44)
SCHEMBL8440146 0.76 KDM4E (0.52) ROCK2ROCK1CDC42BPACDC42BPB
SCHEMBL30336388 0.76 SRC (0.39) ROCK2ROCK1CDC42BPACDC42BPBTSHR
SCHEMBL13174924 0.76 SRC (0.39) ROCK2ROCK1CDC42BPACDC42BPBTSHR
Hydrochloric Acid SCHEMBL8435753 0.74 KDM4E (0.50) ROCK2ROCK1CDC42BPACDC42BPB
Hydrochloric Acid SCHEMBL8438819 0.74 KDM4E (0.50) ROCK2ROCK1CDC42BPACDC42BPB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1930319-B1 Proline derivatives and use thereof as drugs MITSUBISHI TANABE PHARMA CORP (JP) 2012-05-02 EP disclosed