SCHEMBL6127902

SCHEMBL6127902

CN1CCC=C1C(=O)Nc1c(F)cccc1F

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
PDE4D Q08499 3/20 0.40
KMT2A Q03164 1/20 0.40
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
HDAC1 Q13547 1/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
NLRP3 Q96P20 1/20 0.37
NOX1 Q9Y5S8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6127908 0.75 ALDH1A1 (0.43) ALDH1A1PDE4DKMT2APDE4APDE4B
SCHEMBL23808915 0.68 KMT2A (0.63) ALDH1A1KMT2ALMNAHTT
SCHEMBL25422914 0.68 TP53 (0.40) ALDH1A1KMT2AMAPTHTT
SCHEMBL2732129 0.68 RAB9A (0.51) ALDH1A1PDE4DKMT2AHDAC1MAPT
SCHEMBL1430230 0.66 KMT2A (0.55) ALDH1A1PDE4DKMT2AHDAC1NLRP3
SCHEMBL20560667 0.66 KMT2A (0.55) ALDH1A1PDE4DKMT2ANLRP3NOX1
SCHEMBL13182376 0.66
SCHEMBL12283650 0.66
SCHEMBL10173395 0.66 L3MBTL1 (0.40) ALDH1A1KMT2AKDM4E
SCHEMBL2732151 0.66 ALDH1A1 (0.44) ALDH1A1PDE4DKMT2AHDAC1NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012056478-A1 OXAZOLE AND ISOXAZOLE CRAC MODULATORS LUPIN LIMITED (IN) 2012-05-03 WO disclosed