Quinazoline

Quinazoline

SCHEMBL6130196

c1ccc2ncncc2c1.c1cnc2ncncc2n1

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.69
PIK3CD O00329 1/20 0.47
PIK3CA P42336 1/20 0.47
ALDH1A1 P00352 1/20 0.44
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
CYP2A6 P11509 1/20 0.36
METAP2 P50579 1/20 0.36
METAP1 P53582 1/20 0.36
CYP1A2 P05177 2/20 0.35
PIK3CG P48736 1/20 0.35
TDO2 P48775 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL27968729 0.90 ALDH1A1 (0.59) EGFRPIK3CDPIK3CAALDH1A1PDGFRB
Quinoxaline SCHEMBL150387 0.87 EGFR (0.83) EGFRPIK3CDPIK3CAALDH1A1PDGFRB
Acridine SCHEMBL27559723 0.85 ALDH1A1 (0.50) EGFRPIK3CDPIK3CAALDH1A1PDGFRB
Quinazoline SCHEMBL29490398 0.83 EGFR (1.00) EGFRPIK3CDPIK3CAALDH1A1PDGFRB
Quinazoline SCHEMBL29356169 0.83 EGFR (1.00) EGFRPIK3CDPIK3CAALDH1A1PDGFRB
Quinazoline SCHEMBL22833783 0.83 EGFR (1.00) EGFRPIK3CDPIK3CAALDH1A1PDGFRB
Quinazoline SCHEMBL5920 0.83 EGFR (1.00) EGFRPIK3CDPIK3CAALDH1A1PDGFRB
SCHEMBL7000618 0.82 EGFR (0.42) EGFRALDH1A1METAP2METAP1CYP1A2
SCHEMBL29048833 0.82 EGFR (0.41) EGFRPIK3CDPIK3CAALDH1A1CYP2A6
Quinoline SCHEMBL156755 0.82 EGFR (0.80) EGFRPIK3CDPIK3CAALDH1A1PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389909-A4 ANTIMICROBIAL COMPOUNDS AND METHODS FOR THEIR USE OLIGOS ETC INC (US) 2005-03-30 EP disclosed
EP-1389909-A1 ANTIMICROBIAL COMPOUNDS AND METHODS FOR THEIR USE Oligos Etc. Inc. (US) 2004-02-25 EP disclosed
WO-2002089581-A1 ANTIMICROBIAL COMPOUNDS AND METHODS FOR THEIR USE OLIGOS ETC. INC. (US) 2002-11-14 WO disclosed
WO-1999011622-A1 AMINO-SUBSTITUTED COMPOUNDS, METHODS, AND COMPOSITIONS FOR INHIBITING PARP ACTIVITY GUILFORD PHARMACEUTICALS INC. (US) 1999-03-11 WO disclosed