SCHEMBL6131890

SCHEMBL6131890

CN(C)C(=O)Oc1ccc(CN2CCN(c3ccccc3Cl)CC2)cc1F

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
KDM4E B2RXH2 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
MAPK1 P28482 1/20 0.47
HTR7 P34969 3/20 0.46
GAA P10253 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
BCHE P06276 1/20 0.46
MAOA P21397 1/20 0.46
ACHE P22303 1/20 0.46
MAOB P27338 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7690877 0.99 ALDH1A1 (0.51) ALDH1A1KDM4ETDP1MAPK1HTR7
SCHEMBL6131975 0.88 BCHE (0.57) ALDH1A1KDM4ETDP1HTR7BCHE
Hydrochloric Acid SCHEMBL6131817 0.87 BCHE (0.56) ALDH1A1KDM4ETDP1HTR7BCHE
Hydrochloric Acid SCHEMBL6131772 0.87 ALDH1A1 (0.54) ALDH1A1KDM4ETDP1HTR7BCHE
SCHEMBL6131769 0.83 ALDH1A1 (0.67) ALDH1A1KDM4ETDP1MAPK1GAA
SCHEMBL6132073 0.82 ALDH1A1 (0.66) ALDH1A1KDM4ETDP1MAPK1HTR7
SCHEMBL6131832 0.79 KDM4E (0.63) ALDH1A1KDM4EMAPK1HTR7BCHE
SCHEMBL6131998 0.79 KDM4E (0.66) ALDH1A1KDM4ETDP1MAPK1HTR7
Hydrochloric Acid SCHEMBL6131893 0.78 KDM4E (0.62) ALDH1A1KDM4EMAPK1HTR7SMN1; SMN2
SCHEMBL6131790 0.78 ADRA1D (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP claimed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP claimed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO claimed