SCHEMBL6131975

SCHEMBL6131975

COc1cc(CN2CCN(c3ccccc3Cl)CC2)ccc1OC(=O)N(C)C

nearest known ligand 0.69

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.57
MAOA P21397 1/20 0.57
ACHE P22303 1/20 0.57
MAOB P27338 1/20 0.57
ALDH1A1 P00352 4/20 0.55
KDM4E B2RXH2 3/20 0.55
KMT2A Q03164 1/20 0.55
DRD2 P14416 3/20 0.54
ALOX15 P16050 1/20 0.53
TSHR P16473 1/20 0.53
HTR7 P34969 2/20 0.53
TDP1 Q9NUW8 1/20 0.53
DRD4 P21917 2/20 0.53
DRD3 P35462 2/20 0.53
UTS2R Q9UKP6 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6131817 0.99 BCHE (0.56) BCHEMAOAACHEMAOBALDH1A1
Hydrochloric Acid SCHEMBL6131772 0.95 ALDH1A1 (0.54) BCHEMAOAACHEMAOBALDH1A1
SCHEMBL6131832 0.92 KDM4E (0.63) BCHEMAOAACHEMAOBALDH1A1
Hydrochloric Acid SCHEMBL6131893 0.91 KDM4E (0.62) BCHEMAOAACHEMAOBALDH1A1
SCHEMBL6131790 0.90 ADRA1D (0.57) KMT2ADRD2DRD4DRD3
SCHEMBL6131962 0.90 KDM4E (0.62) BCHEMAOAACHEMAOBALDH1A1
SCHEMBL6131998 0.90 KDM4E (0.66) ALDH1A1KDM4EKMT2ADRD2ALOX15
SCHEMBL6131769 0.89 ALDH1A1 (0.67) BCHEMAOAACHEMAOBALDH1A1
Hydrochloric Acid SCHEMBL6131814 0.89 KDM4E (0.61) BCHEMAOAACHEMAOBALDH1A1
SCHEMBL6131890 0.88 ALDH1A1 (0.52) BCHEMAOAACHEMAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP claimed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP claimed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO claimed