SCHEMBL6132002

SCHEMBL6132002

COc1cc(CN2CCN(c3ccccc3F)CC2)ccc1OC(=O)N1CCc2ccccc2C1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.60
ALDH1A1 P00352 8/20 0.60
TDP1 Q9NUW8 2/20 0.60
GAA P10253 3/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
ALOX15 P16050 2/20 0.54
POLB P06746 1/20 0.54
MAPK1 P28482 1/20 0.54
KMT2A Q03164 2/20 0.51
MAPT P10636 2/20 0.51
MEN1 O00255 1/20 0.51
DRD2 P14416 2/20 0.49
HTR1A P08908 1/20 0.49
DRD4 P21917 1/20 0.48
DRD3 P35462 1/20 0.48
ACHE P22303 1/20 0.48
HTT P42858 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
TAAR1 Q96RJ0 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7687618 0.99 KDM4E (0.59) KDM4EALDH1A1TDP1GAASMN1; SMN2
SCHEMBL6132069 0.83 ALDH1A1 (0.58) KDM4EALDH1A1SMN1; SMN2MAPK1KMT2A
SCHEMBL6131795 0.81 ALDH1A1 (0.67) KDM4EALDH1A1TDP1GAASMN1; SMN2
SCHEMBL6131769 0.81 ALDH1A1 (0.67) KDM4EALDH1A1TDP1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL6131911 0.79 ALDH1A1 (0.65) KDM4EALDH1A1TDP1GAASMN1; SMN2
SCHEMBL6131807 0.76 ALDH1A1 (0.61) KDM4EALDH1A1TDP1GAASMN1; SMN2
SCHEMBL6131806 0.75 ALDH1A1 (0.60) KDM4EALDH1A1TDP1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL6131845 0.75 ALDH1A1 (0.60) KDM4EALDH1A1TDP1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL6131844 0.75 ALDH1A1 (0.59) KDM4EALDH1A1TDP1GAASMN1; SMN2
SCHEMBL10414099 0.74 USP2 (0.65) KDM4EALDH1A1TDP1GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP claimed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP claimed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO claimed