SCHEMBL6131806

SCHEMBL6131806

COc1cc(CN2CCN(c3ccccc3F)CC2)ccc1OC(=O)NC(C)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.60
KDM4E B2RXH2 8/20 0.58
TDP1 Q9NUW8 2/20 0.58
GAA P10253 3/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
ALOX15 P16050 3/20 0.54
POLB P06746 1/20 0.54
MAPK1 P28482 1/20 0.54
KMT2A Q03164 4/20 0.48
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
DRD3 P35462 1/20 0.48
TSHR P16473 2/20 0.47
LMNA P02545 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
FAAH O00519 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6131844 0.99 ALDH1A1 (0.59) ALDH1A1KDM4ETDP1GAASMN1; SMN2
SCHEMBL6131795 0.86 ALDH1A1 (0.67) ALDH1A1KDM4ETDP1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL6131911 0.84 ALDH1A1 (0.65) ALDH1A1KDM4ETDP1GAASMN1; SMN2
SCHEMBL6131769 0.82 ALDH1A1 (0.67) ALDH1A1KDM4ETDP1GAASMN1; SMN2
SCHEMBL6131807 0.80 ALDH1A1 (0.61) ALDH1A1KDM4ETDP1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL6131845 0.79 ALDH1A1 (0.60) ALDH1A1KDM4ETDP1GAASMN1; SMN2
SCHEMBL6131943 0.77 KDM4E (0.63) ALDH1A1KDM4ETDP1SMN1; SMN2ALOX15
SCHEMBL6131799 0.77 ADRA1D (0.56) ALDH1A1KDM4ETDP1GAASMN1; SMN2
SCHEMBL6131777 0.76 ADRA1D (0.59) ALDH1A1KDM4ETDP1GAASMN1; SMN2
SCHEMBL6131830 0.76 KDM4E (0.62) ALDH1A1KDM4ETDP1GAAALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP claimed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP claimed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO claimed