Bromide

Bromide

SCHEMBL6132084

Br.C#CCOc1cc(CN2CCCCC2)ccc1OC

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIGMAR1 known ✓ Q99720 1/20 0.46
DRD2 P14416 1/20 0.61
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
GAA P10253 1/20 0.51
MAPK1 P28482 1/20 0.50
HSD17B10 Q99714 1/20 0.50
POLB P06746 1/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6131905 0.99 DRD2 (0.63) DRD2KMT2AMEN1GAAMAPK1
SCHEMBL7680831 0.97 DRD2 (0.64) DRD2KMT2AMEN1GAAMAPK1
Hydrochloric Acid SCHEMBL6132064 0.96 DRD2 (0.63) DRD2KMT2AMEN1GAAMAPK1
SCHEMBL5667128 0.87 DRD2 (0.65) DRD2KMT2AMEN1MAPK1HSD17B10
SCHEMBL6131946 0.86 HTT (0.61) DRD2KMT2AMEN1MAPK1HSD17B10
Hydrochloric Acid SCHEMBL5667186 0.86 DRD2 (0.64) DRD2KMT2AMEN1MAPK1HSD17B10
SCHEMBL6131868 0.84 MAPK1 (0.52) DRD2KMT2AMEN1GAAMAPK1
SCHEMBL28191613 0.83 GAA (0.66) KMT2AMEN1GAAMAPK1SIGMAR1
SCHEMBL16884151 0.82 GAA (0.63) KMT2AMEN1GAAMAPK1SIGMAR1
SCHEMBL7688903 0.80 KDM4E (0.53) DRD2KMT2AMEN1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed