SCHEMBL6134547

SCHEMBL6134547

CC(C)n1nc(C(=CN(C)C)C(=O)c2cccc(F)c2)ccc1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.40
CES1 P23141 2/20 0.40
CHRNB2 P17787 1/20 0.35
SLC6A2 P23975 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HPGD P15428 2/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
KDM4E B2RXH2 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRL1 P41146 1/20 0.33
PARP1 P09874 1/20 0.33
HDAC6 Q9UBN7 2/20 0.32
PIK3CD O00329 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6134543 1.00 CES2 (0.40) CES2CES1CHRNB2SLC6A2CHRNB4
SCHEMBL6133324 0.87 POLB (0.43) CHRNB2SLC6A2CHRNB4CHRNA3CHRNA4
SCHEMBL6133325 0.87 POLB (0.43) CHRNB2SLC6A2CHRNB4CHRNA3CHRNA4
SCHEMBL6133710 0.87 CYP1A2 (0.35) CES2CES1ALDH1A1PKMMAPT
SCHEMBL6133711 0.87 CYP1A2 (0.35) CES2CES1ALDH1A1PKMMAPT
SCHEMBL6135115 0.87 CES2 (0.43) CES2ALDH1A1OPRM1OPRL1HDAC6
SCHEMBL6135116 0.87 CES2 (0.43) CES2ALDH1A1OPRM1OPRL1HDAC6
SCHEMBL6134296 0.87 LMNA (0.40) CES2CES1HPGDALDH1A1PKM
SCHEMBL6134293 0.87 LMNA (0.40) CES2CES1HPGDALDH1A1PKM
SCHEMBL6133458 0.81 CYP11B1 (0.40) CES2CES1HPGDALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050043315-A1 Aminopyrimidine compounds, processes for their preparation and pharmaceutical compositions containing them ASTELLAS PHARMA INC. (JP) 2005-02-24 US disclosed
WO-2003057689-A1 AMINOPYRIMIDINE COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-07-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050043315-A1 Aminopyrimidine compounds, processes for their preparation and pharmaceutical compositions containing them ADORA2B, ADORA2A, ADORA1 CES2 4034/4885CES1 3947/4885CHRNB2 182/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.