SCHEMBL6134889

SCHEMBL6134889

CC(C)n1nc(-c2cnc(N)nc2-c2c(Cl)cccc2Cl)ccc1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 4/20 0.42
SRC P12931 4/20 0.42
EGFR P00533 2/20 0.42
FGFR2 P21802 2/20 0.42
FGFR4 P22455 2/20 0.42
FGFR3 P22607 2/20 0.42
MDM2 Q00987 2/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
PRKD3 O94806 1/20 0.35
PRKCG P05129 1/20 0.35
PRKCB P05771 1/20 0.35
PDGFRB P09619 1/20 0.35
PDGFRA P16234 1/20 0.35
PRKCA P17252 1/20 0.35
PRKCH P24723 1/20 0.35
MAPK3 P27361 1/20 0.35
MAPK1 P28482 1/20 0.35
PRKCI P41743 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6134855 0.89 KDM5B (0.36) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL6134198 0.89 FGFR1 (0.39) FGFR1SRCEGFRFGFR2FGFR4
SCHEMBL6133980 0.87 ADORA1 (0.35) FGFR1SRCFGFR2FGFR3MDM2
SCHEMBL6135304 0.85 ADORA1 (0.40) FGFR1SRCEGFRFGFR2FGFR3
SCHEMBL6134599 0.84 ADORA1 (0.53) SRCADORA2AADORA2BADORA1
SCHEMBL6134188 0.83 LMNA (0.45) ADORA2AADORA2BADORA1
SCHEMBL6134324 0.83 ADORA1 (0.47) ADORA2AADORA2BADORA1
SCHEMBL6134367 0.83 ADORA1 (0.50) FGFR1SRCEGFRFGFR2FGFR3
SCHEMBL6134252 0.81 ADORA2A (0.38) FGFR1SRCFGFR2FGFR3ADORA2A
SCHEMBL6133385 0.81 ADORA1 (0.54) SRCADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050043315-A1 Aminopyrimidine compounds, processes for their preparation and pharmaceutical compositions containing them ASTELLAS PHARMA INC. (JP) 2005-02-24 US disclosed
WO-2003057689-A1 AMINOPYRIMIDINE COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-07-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050043315-A1 Aminopyrimidine compounds, processes for their preparation and pharmaceutical compositions containing them ADORA2B, ADORA2A, ADORA1 FGFR1 3416/4885SRC 2622/4885EGFR 2577/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.