SCHEMBL6140901

SCHEMBL6140901

CN(C)CCNc1ccc(CC=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.41
RAD52 P43351 1/20 0.39
SIGMAR1 Q99720 2/20 0.38
LMNA P02545 2/20 0.38
CYP1A2 P05177 1/20 0.38
MAOA P21397 1/20 0.38
CNR1 P21554 1/20 0.38
DRD4 P21917 1/20 0.38
ACHE P22303 1/20 0.38
HRH2 P25021 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
MAPK1 P28482 1/20 0.38
NTSR1 P30989 1/20 0.38
HRH1 P35367 1/20 0.38
DRD3 P35462 1/20 0.38
SCN1A P35498 1/20 0.38
HTR2B P41595 1/20 0.38
SCN7A Q01118 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6439791 0.90 LMNA (0.43) HRH3SIGMAR1LMNACYP1A2MAOA
SCHEMBL6141318 0.80 NOS1 (0.50) RAD52CYP1A2MALT1CYP2C19CACNA1B
SCHEMBL3694813 0.80 CYP2A6 (0.44) HRH3RAD52SIGMAR1LMNACYP1A2
SCHEMBL15613318 0.79 HPGD (0.47) HRH3SIGMAR1LMNACYP1A2MAOA
SCHEMBL250769 0.78 KEAP1 (0.49) HRH3CYP2C19CACNA1BNOS1NOS2
SCHEMBL249718 0.76 CACNA1B (0.43) HRH3KDM4ECYP2C19CACNA1BNOS1
SCHEMBL4037295 0.76 MAPT (0.35) DRD4MAPT
SCHEMBL23928190 0.75 HRH3 (0.45) HRH3CYP1A2HTR2AKDM4ECYP2C19
SCHEMBL81430 0.75 MAPT (0.67) HRH3RAD52MAPK1KDM4EBLM
SCHEMBL10053347 0.75 MAPT (0.47) LMNAMAPK1KDM4EBLMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1515940-A2 AMINOALKOXY-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-03-23 EP disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed
WO-2003097574-A2 AMINOALKOXY-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed