SCHEMBL6148010

SCHEMBL6148010

NS(=O)(=O)CCCC(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 1/20 0.37
CA7 P43166 1/20 0.36
CA13 Q8N1Q1 1/20 0.36
ARG1 P05089 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1933559 0.83 CA1 (0.40) CA1CA2CA9CA7CA13
SCHEMBL309951 0.78 CES1 (0.33)
SCHEMBL353498 0.76 ESR1 (0.32)
SCHEMBL216634 0.74 APP (0.46)
SCHEMBL14814813 0.74 ALDH1A1 (0.35)
SCHEMBL7204059 0.74 CA2 (0.33) CA2ARG1
SCHEMBL14814810 0.74
SCHEMBL3097818 0.74
SCHEMBL10457263 0.73 CA2 (0.43) CA1CA2CA9CA7
SCHEMBL10405537 0.73 CA2 (0.39) CA1CA2CA9CA7ARG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019046465-A2 THERAPEUTIC INDOLES RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2019-03-07 WO claimed
US-10392348-B2 2-oxo-3,4-dihydroquinoline compounds as plant growth regulators SYNGENTA PARTICIPATIONS AG (CH) 2019-08-27 US disclosed
WO-2019046465-A2 THERAPEUTIC INDOLES RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2019-03-07 WO disclosed
US-20180044297-A1 2-OXO-3,4-DIHYDROQUINOLINE COMPOUNDS AS PLANT GROWTH REGULATORS SYNGENTA PARTICIPATIONS AG (CH) 2018-02-15 US disclosed
CN-101177385-B Aryl sulfonic acid amides and analogues as well as its purpose in curing neural degeneration disease BAYER AG 2011-06-15 CN disclosed
CN-100453529-C Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases BAYER AG (DE) 2009-01-21 CN disclosed
CN-101177385-A Aryl sulfonic acid amides and analogues as well as its purpose in curing neural degeneration disease BAYER AG (DE) 2008-05-14 CN disclosed
CN-100371318-C Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases BAYER AG (DE) 2008-02-27 CN disclosed
CN-1754873-A Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases BAYER AG (DE) 2006-04-05 CN disclosed
EP-1105370-B9 NOVEL ARYL SULPHONAMIDES AND ANALOGUES BAYER HEALTHCARE AG (DE) 2005-01-12 EP disclosed
US-6573278-B2 For therapy and prophylaxis of cerebral apoplexy and craniocerebral trauma BAYER AKTIENGESELLSCHAFT (DE) 2003-06-03 US disclosed
US-20030073727-A1 Novel arylsulphonamides and analogues MITTENDORF JOACHIM (DE) 2003-04-17 US disclosed
US-6545050-B1 Prophylaxis and treatment of neurodegenerative disorders, in particular for the treatment of cerebral apoplexy, craniocerebral trauma, pain and spasticity. BAYER AKTIENGESELLSCHAFT (DE) 2003-04-08 US disclosed
EP-0966436-B1 ARYL SULFONAMIDES AND ANALOGUES THEREOF AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES BAYER AG (DE) 2002-12-11 EP disclosed
US-6469054-B1 PROPHYLAXIS AND TREATMENT OF NEURODEGENERATIVE DISORDERS, IN PARTICULAR FOR THE TREATMENT OF CEREBRAL APOPLEXY, CRANIOCEREBRAL TRAUMA, PAIN AND SPASTICITY BAYER AKTIENGESELLSHAFT (DE) 2002-10-22 US disclosed
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
US-20020072529-A1 Arylsulfonamides and analogues BAYER INTELLECTUAL PROPERTY GMBH (DE) 2002-06-13 US disclosed
US-6262112-B1 1-(4,4,4-TRIFLUOROBUTYLSULPHONYLOXY)-3-(2-(HYDROXYMETHYL)INDAN -4-YLOXY)-BENZENE BAYER AKTIENGESELLSCHAFT (DE) 2001-07-17 US disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed
CN-1253545-A Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases BAYER AG (DE) 2000-05-17 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10392348-B2 2-oxo-3,4-dihydroquinoline compounds as plant growth regulators CDC25B, OSR1, CDC25C CA1 4131/4885CA2 1966/4885CA9 4525/4885
US-20030073727-A1 Novel arylsulphonamides and analogues PRSS12, OPRL1, CTSH CA1 4138/4885CA2 4123/4885CA9 4576/4885
US-20180044297-A1 2-OXO-3,4-DIHYDROQUINOLINE COMPOUNDS AS PLANT GROWTH REGULATORS CDC25B, OSR1, CDC25C CA1 4131/4885CA2 1966/4885CA9 4525/4885
US-20020072529-A1 Arylsulfonamides and analogues ARSA, PRSS12, SNCA CA1 1982/4885CA2 3918/4885CA9 3161/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.