SCHEMBL6152662

SCHEMBL6152662

C=CC(=O)ONC(=O)CC(C)=O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 7/20 0.36
HPGD P15428 1/20 0.35
ALDH1A1 P00352 7/20 0.35
MGAM O43451 1/20 0.34
GAA P10253 1/20 0.34
SI P14410 1/20 0.34
MGAM2 Q2M2H8 1/20 0.34
TP53 P04637 3/20 0.34
HIF1A Q16665 3/20 0.34
CYP3A4 P08684 2/20 0.34
HSD17B10 Q99714 1/20 0.34
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
THRB P10828 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28817744 0.83 TSHR (0.37) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL28220847 0.81 TSHR (0.41) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL5741244 0.78
SCHEMBL28838342 0.78 CTSD (0.45) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL20996194 0.77 ALDH1A1 (0.36) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL979061 0.74 ALDH1A1 (0.38) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL6153042 0.74 ALDH1A1 (0.48) TSHRALDH1A1MGAMGAASI
SCHEMBL2707512 0.73 TSHR (0.33) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL14798439 0.73 PHF8 (0.45) TSHRALDH1A1TP53HIF1ACYP3A4
SCHEMBL29065557 0.73 HCAR2 (0.50) ALDH1A1MGAMGAASIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986611-B1 CROSS-LINKABLE SURFACE COATINGS AND PROCESS OF PREPARATION JOHNSON POLYMER LLC (US) 2005-01-26 EP disclosed
US-6090882-A Crosslinkable surface coatings and process of preparation S. C. JOHNSON COMMERCIAL MARKETS, INC. (US) 2000-07-18 US disclosed
EP-0873303-B1 ETHYLENICALLY-UNSATURED 1,3-DIKETOAMIDE FUNCTIONAL COMPOUNDS, POLYMERS THEREOF AND LATEX FORMULATIONS CONTAINING THE SAME JOHNSON S C COMM MARKETS INC (US) 2000-05-03 EP disclosed
EP-0986611-A1 CROSS-LINKABLE SURFACE COATINGS AND PROCESS OF PREPARATION S.C. Johnson Commercial Markets, Inc. (US) 2000-03-22 EP disclosed
US-5889098-A A LATEX FORMULATION COMPRISES 1,3-DIKETOAMIDE PENDANT GROUP DERIVED FROM AN ETHYLENICALLY UNSATURATED 1,3-DIKETOAMIDE FUNCTIONAL COMPOUND, A POLYFUNCTIONAL AMINE AND AN EVAPORABLE AQUEOUS CARRIER; CROSSLINKABLE; STORAGE STABILITY S. C. JOHNSON COMMERCIAL MARKETS, INC. (US) 1999-03-30 US disclosed
US-5886116-A HYDROLYTIC STABILITY S.C. JOHNSON COMMERCIAL MARKETS, INC. (US) 1999-03-23 US disclosed
US-5872297-A Ethylenically-unsaturated 1,3-diketoamide functional compounds S. C. JOHNSON COMMERCIAL MARKETS, INC. (US) 1999-02-16 US disclosed
WO-1998054256-A1 CROSS-LINKABLE SURFACE COATINGS AND PROCESS OF PREPARATION S. C. JOHNSON COMMERCIAL MARKETS, INC. (US) 1998-12-03 WO disclosed
EP-0873303-A1 ETHYLENICALLY-UNSATURED 1,3-DIKETOAMIDE FUNCTIONAL COMPOUNDS, POLYMERS THEREOF AND LATEX FORMULATIONS CONTAINING THE SAME S.C.JOHNSON & SON, INC. (US) 1998-10-28 EP disclosed
WO-1997008134-A1 ETHYLENICALLY-UNSATURATED 1,3-DIKETOAMIDE FUNCTIONAL COMPOUNDS, POLYMERS THEREOF AND LATEX FORMULATIONS CONTAINING THE SAME S.C. JOHNSON & SON, INC. (US) 1997-03-06 WO disclosed