SCHEMBL6152773

SCHEMBL6152773

C=CC(=O)c1cccc(-n2nnnc2S)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.46
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
POLB P06746 3/20 0.41
HPGD P15428 2/20 0.41
AKT1 P31749 1/20 0.40
CPB1 P15086 1/20 0.39
LMNA P02545 2/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPT P10636 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
KDM4E B2RXH2 1/20 0.38
EGFR P00533 1/20 0.38
CYP3A4 P08684 1/20 0.38
PKM P14618 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10467466 0.84 TP53 (0.46) TP53KMT2AMEN1POLBHPGD
SCHEMBL8021678 0.83 TP53 (0.60) TP53KMT2AMEN1POLBHPGD
SCHEMBL14498646 0.82 TP53 (0.49) TP53KMT2AMEN1POLBHPGD
SCHEMBL13297855 0.80 HDAC8 (0.45) TP53KMT2AMEN1POLBHPGD
SCHEMBL8943869 0.78 TP53 (0.46) TP53KMT2AMEN1POLBHPGD
SCHEMBL13297724 0.78 AOC2 (0.54) TP53KMT2AMEN1POLBHPGD
SCHEMBL11563751 0.78 TGM2 (0.48) LMNAL3MBTL1ALDH1A1MAPTEGFR
SCHEMBL6153223 0.75 MAPK1 (0.53) TP53KMT2AMEN1POLBHPGD
SCHEMBL10505126 0.75 TP53 (0.49) TP53KMT2ALMNASMN1; SMN2ALDH1A1
SCHEMBL14498645 0.75 TP53 (0.49) TP53KMT2AMEN1POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-H963-H Containing development inhibitor and reducible dye FUJI PHOTO FILM CO., LTD. (JP) 1991-09-03 US claimed
EP-1037106-B1 Color diffusion transfer photographic material FUJI PHOTO FILM CO LTD (JP) 2005-01-26 EP disclosed
US-6376164-B1 CONTAINING 2-THIOBENZOTHIAZOLE COMPOUND FUJI PHOTO FILM CO., LTD. (JP) 2002-04-23 US disclosed
US-6187527-B1 A SENSITIVITY REGULATION BY PROLONGING THE BLACK AND WHITE DEVELOPMENT TIME DURING COLOR REVERSAL PROCESS IS CONDUCTED IN ORDER TO COMPENSATE FOR ANY UNDER-EXPOSURE OF A COLOR PHOTOGRAPHIC LIGHTSENSITIVE MATERIAL. FUJI PHOTO FILM CO., LTD. (JP) 2001-02-13 US disclosed
EP-1037106-A1 Color diffusion transfer photographic material FUJI PHOTO FILM CO., LTD. (JP) 2000-09-20 EP disclosed
US-6013421-A EXPOSURE TO LIGHT FOR SILVER HALIDE EMULSIONS FOR COLOR PHOTOGRAPHY FUJI PHOTO FILM CO., LTD. (JP) 2000-01-11 US disclosed
EP-0534283-B1 Silver halide photographic light-sensitive material FUJI PHOTO FILM CO LTD (JP) 1997-12-17 EP disclosed
US-5691125-A CYAN DYE-FORMING COUPLER, STORAGE STABLE FUJI PHOTO FILM CO., LTD. (JP) 1997-11-25 US disclosed
US-5609999-A INDOLE DYE; STORAGE STABILITY, COLOR REPRODUCIBILITY, SHARPNESS FUJI PHOTO FILM CO., LTD. (JP) 1997-03-11 US disclosed
EP-0537659-B1 Silver halide color photographic light-sensitive material, and method of processing the same FUJI PHOTO FILM CO LTD (JP) 1997-01-15 EP disclosed
US-4886736-A COUPLERS AND COMPOUND CAPABLE OF RELEASING PHOTOGRAPHICALLY USEFUL GROUP UPON REDUCTION FUJI PHOTO FILM CO., LTD. (JP) 1989-12-12 US disclosed
EP-0167168-B1 SILVER HALIDE PHOTOGRAPHIC MATERIAL FUJI PHOTO FILM CO., LTD. (JP) 1989-11-15 EP disclosed
EP-0198438-B1 SILVER HALIDE PHOTOGRAPHIC LIGHT-SENSITIVE MATERIAL FUJI PHOTO FILM CO., LTD. (JP) 1989-10-18 EP disclosed
US-4840887-A USEFUL GROUP RELEASED BY CLEAVAGE BETWEEN SULFONYL GROUP AND A NITROGEN, SULFUR OR OXYGEN ATOM; STABILITY FUJI PHOTO FILM CO., LTD. (JP) 1989-06-20 US disclosed
US-4820622-A RELEASING DIFFUSIBLE DYE IN ALKALINE SYSTEM AFTER HALIDE REDUCTION FUJI PHOTO FILM CO., LTD. (JP) 1989-04-11 US disclosed
US-4783396-A Silver halide photographic materials FUJI PHOTO FILM CO., LTD. (JP) 1988-11-08 US disclosed
US-4770990-A Silver halide photographic light-sensitive material containing a compound capable of imagewise releasing a photographically useful group during development FUJI PHOTO FILM CO., LTD. (JP) 1988-09-13 US disclosed
EP-0220746-A2 Silver halide photographic materials FUJI PHOTO FILM CO., LTD. (JP) 1987-05-06 EP disclosed
EP-0198438-A2 Silver halide photographic light-sensitive material FUJI PHOTO FILM CO., LTD. (JP) 1986-10-22 EP disclosed
EP-0167168-A2 Silver halide photographic material FUJI PHOTO FILM CO., LTD. (JP) 1986-01-08 EP disclosed