SCHEMBL6153422

SCHEMBL6153422

Nc1cccc(-c2ccc(OCCN3CCN(CCc4ccccc4)CC3)c3c2C2CCC3CC2)n1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 18/20 0.60
NOS3 P29474 17/20 0.60
NOS2 P35228 12/20 0.60
CHRM2 P08172 1/20 0.44
CHRM4 P08173 1/20 0.44
DRD2 P14416 1/20 0.42
HTR2A P28223 1/20 0.42
HTR7 P34969 1/20 0.42
ADRA1A P35348 1/20 0.42
HTR6 P50406 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6152955 0.89 NOS3 (0.72) NOS1NOS3NOS2
SCHEMBL6152196 0.88 NOS3 (0.69) NOS1NOS3NOS2
SCHEMBL6153424 0.86 NOS1 (0.50) NOS1NOS3NOS2CHRM2CHRM4
SCHEMBL6152435 0.85 NOS3 (0.69) NOS1NOS3NOS2
SCHEMBL5833437 0.85 NOS1 (0.78) NOS1NOS3NOS2CHRM2CHRM4
SCHEMBL5833985 0.84 NOS3 (0.69) NOS1NOS3NOS2
SCHEMBL6153425 0.83 NOS3 (0.56) NOS1NOS3NOS2DRD2HTR2A
SCHEMBL5833190 0.82 NOS1 (0.79) NOS1NOS3NOS2CHRM2CHRM4
SCHEMBL255330 0.80 NOS1 (0.57) NOS1NOS3NOS2CHRM2CHRM4
SCHEMBL6153070 0.80 NOS1 (0.75) NOS1NOS3NOS2DRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1084109-B1 2-AMINOPYRIDINES CONTAINING FUSED RING SUBSTITUENTS AS NITRIC OXIDE SYNTHASE INHIBITORS PFIZER PROD INC (US) 2005-01-26 EP disclosed