SCHEMBL6153424

SCHEMBL6153424

CC(Oc1ccc(-c2cccc(N)n2)c2c1C1CCC2CC1)N1CCN(CCc2ccccc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 18/20 0.50
NOS3 P29474 17/20 0.50
NOS2 P35228 11/20 0.46
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
HTR2A P28223 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6153422 0.86 NOS1 (0.60) NOS1NOS3NOS2CHRM2CHRM4
SCHEMBL6153197 0.86 NOS1 (0.50) NOS1NOS3NOS2
SCHEMBL5833188 0.83 NOS1 (0.58) NOS1NOS3NOS2CHRM2CHRM4
SCHEMBL6699624 0.76 NOS1 (0.60) NOS1NOS3NOS2CHRM2CHRM4
SCHEMBL6152955 0.75 NOS3 (0.72) NOS1NOS3NOS2
SCHEMBL6699620 0.75 NOS1 (0.52) NOS1NOS3NOS2CHRM2CHRM4
SCHEMBL6702757 0.75 NOS1 (0.49) NOS1NOS3NOS2CHRM2CHRM4
SCHEMBL6152196 0.74 NOS3 (0.69) NOS1NOS3NOS2
SCHEMBL7483824 0.74 NOS1 (0.53) NOS1NOS3NOS2CHRM2CHRM4
SCHEMBL6703557 0.73 NOS1 (0.48) NOS1NOS3NOS2CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1084109-B1 2-AMINOPYRIDINES CONTAINING FUSED RING SUBSTITUENTS AS NITRIC OXIDE SYNTHASE INHIBITORS PFIZER PROD INC (US) 2005-01-26 EP disclosed