SCHEMBL6153818

SCHEMBL6153818

NC(=O)c1ccc(NC(=O)C2CCC(CNC(=O)O)CC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.54
RAB9A P51151 1/20 0.51
KMT2A Q03164 5/20 0.49
MEN1 O00255 3/20 0.49
LMNA P02545 1/20 0.49
MAPT P10636 4/20 0.48
GAA P10253 1/20 0.48
GFER P55789 1/20 0.48
CYP2C9 P11712 1/20 0.47
HPGD P15428 1/20 0.47
NAMPT P43490 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25845705 0.84 NAMPT (0.62) RAB9AKMT2AMEN1LMNAMAPT
SCHEMBL6154809 0.83 KMT2A (0.54) RAB9AKMT2AMEN1LMNAMAPT
SCHEMBL6154813 0.83 KMT2A (0.54) RAB9AKMT2AMEN1LMNAMAPT
SCHEMBL6153470 0.79 NAMPT (0.56) RAB9AKMT2AMEN1LMNAMAPT
SCHEMBL10618264 0.77 KMT2A (0.56) RAB9AKMT2AMEN1LMNAMAPT
SCHEMBL10618261 0.77 KMT2A (0.56) RAB9AKMT2AMEN1LMNAMAPT
SCHEMBL28241421 0.77 PTPN1 (0.70) RAB9AKMT2AMEN1LMNAMAPT
Hydrochloric Acid SCHEMBL10606970 0.76 KMT2A (0.55) RAB9AKMT2AMEN1LMNAMAPT
Hydrochloric Acid SCHEMBL10606963 0.76 KMT2A (0.55) RAB9AKMT2AMEN1LMNAMAPT
SCHEMBL6153241 0.75 SIRT2 (0.64) RAB9AKMT2AMEN1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050182040-A1 Benzamide derivatives DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2005-08-18 US disclosed
EP-1500643-A1 BENZAMIDE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2005-01-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050182040-A1 Benzamide derivatives ROCK1, ROCK2, NHERF1 MAPK14 43/4885RAB9A 568/4885KMT2A 1307/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.