SCHEMBL6156056

SCHEMBL6156056

[O]CC(=O)NCc1ccccc1C(=O)NCCc1cc(O)c(O)c(O)c1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC6A5 Q9Y345 15/20 0.47
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
ESRRG P62508 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6156568 0.80 CA1 (0.64)
SCHEMBL6264342 0.79 HPGD (0.49) SLC6A5
SCHEMBL6267497 0.75 HPGD (0.51) SLC6A5NPC1RAB9A
SCHEMBL6157584 0.73 KCNA5 (0.43) SLC6A5NPC1RAB9A
SCHEMBL6266482 0.72 KMT2A (0.43) SLC6A5
SCHEMBL31241193 0.70 ESRRG (0.48) NPC1RAB9AESRRG
SCHEMBL31241194 0.70 ESRRG (0.48) NPC1RAB9AESRRG
SCHEMBL6156971 0.70 MAPK8 (0.43) NPC1RAB9A
SCHEMBL6267859 0.69 HPGD (0.47)
SCHEMBL5422657 0.68 TACR1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501813-A2 BENZOTHIADIAZEPINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Astrazeneca AB (SE) 2005-02-02 EP claimed
WO-2003091232-A2 BENZOTHIADIAZEPINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ASTRAZENECA AB (SE) 2003-11-06 WO claimed