SCHEMBL6156568

SCHEMBL6156568

NS(=O)(=O)c1ccc(CCNC(=O)c2ccccc2CNC(=O)C[O])cc1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.64
CA2 P00918 6/20 0.64
CA9 Q16790 4/20 0.64
ALDH1A1 P00352 4/20 0.60
LMNA P02545 1/20 0.60
CA12 O43570 2/20 0.60
KMT2A Q03164 4/20 0.58
GAA P10253 1/20 0.56
HSD17B10 Q99714 1/20 0.55
POLB P06746 1/20 0.55
CA5A P35218 1/20 0.55
CA7 P43166 1/20 0.55
CA5B Q9Y2D0 1/20 0.55
MEN1 O00255 2/20 0.55
RXFP1 Q9HBX9 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6156056 0.80 SLC6A5 (0.47)
SCHEMBL11880873 0.79 CA1 (0.74) CA1CA2CA9ALDH1A1LMNA
SCHEMBL28574459 0.78 ALDH1A1 (0.73) CA1CA2CA9ALDH1A1LMNA
SCHEMBL29609330 0.78 KMT2A (0.73) CA1CA2CA9ALDH1A1LMNA
SCHEMBL30165930 0.76 CA2 (0.70) CA1CA2CA9ALDH1A1LMNA
SCHEMBL28573216 0.76 CA2 (0.70) CA1CA2CA9ALDH1A1LMNA
SCHEMBL6264342 0.76 HPGD (0.49) ALDH1A1LMNAKMT2AGAAMEN1
SCHEMBL29385160 0.75 ALDH1A1 (0.79) CA1CA2CA9ALDH1A1LMNA
SCHEMBL28568182 0.75 ALDH1A1 (0.79) CA1CA2CA9ALDH1A1LMNA
SCHEMBL6046379 0.75 MEN1 (0.90) CA1CA2CA9CA12KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501813-A2 BENZOTHIADIAZEPINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Astrazeneca AB (SE) 2005-02-02 EP disclosed
WO-2003091232-A2 BENZOTHIADIAZEPINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ASTRAZENECA AB (SE) 2003-11-06 WO disclosed