SCHEMBL6157872

SCHEMBL6157872

O=C1CCC(S)C(=O)N1Cc1ccc(Oc2ccc(Br)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.38
HCRTR2 O43614 3/20 0.38
POLB P06746 1/20 0.36
CXCR3 P49682 2/20 0.36
MT-CO2 P00403 1/20 0.36
ALOX5 P09917 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
LTA4H P09960 1/20 0.35
PTGS2 P35354 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
MAPT P10636 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
ACHE P22303 1/20 0.35
SRD5A2 P31213 1/20 0.35
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159504 0.88 HCRTR1 (0.49) HCRTR1HCRTR2POLBMT-CO2ALOX5
SCHEMBL6159715 0.86 HCRTR1 (0.41) HCRTR1HCRTR2POLBCXCR3MT-CO2
SCHEMBL6158749 0.78 HTT (0.37) HCRTR1HCRTR2POLBCXCR3HDAC1
SCHEMBL6159751 0.75 HCRTR1 (0.52) HCRTR1HCRTR2POLBMT-CO2ALOX5
SCHEMBL7082507 0.75 ALDH1A1 (0.48) HCRTR1HCRTR2POLBMT-CO2ALOX5
SCHEMBL6157379 0.75 ALDH1A1 (0.48) HCRTR1HCRTR2POLBMT-CO2ALOX5
SCHEMBL30643636 0.74 CMA1 (0.47) POLBCXCR3MAPT
SCHEMBL6160031 0.73 HCRTR1 (0.49) HCRTR1HCRTR2POLBMT-CO2ALOX5
SCHEMBL5767794 0.72 CA12 (0.58) POLBHDAC1HDAC8HDAC6CHRM5
Bromide SCHEMBL6161403 0.72 HCRTR1 (0.48) HCRTR1HCRTR2POLBMT-CO2ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-20040157894-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-08-12 US disclosed
US-6699881-B2 MATRIX METALLOPROTEASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-03-02 US disclosed
US-20030078253-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2003-04-24 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-1132379-A1 NOVEL THIOL DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND UTILIZATION THEREOF Takeda Chemical Industries, Ltd. (JP) 2001-09-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078253-A1 Thiol compounds, their production and use TST, QSOX1, SULT1E1 HCRTR1 1949/4885HCRTR2 1842/4885POLB 3567/4885
US-20040157894-A1 Thiol compounds, their production and use TST, SULT1E1, QSOX1 HCRTR1 1930/4885HCRTR2 1754/4885POLB 3489/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.