SCHEMBL6158970

SCHEMBL6158970

COc1cc(C(CCN)CCCc2cccnc2)cc(OC)c1OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.48
PTAFR P25105 5/20 0.47
HRH1 P35367 2/20 0.46
FKBP1A P62942 5/20 0.44
ABCC1 P33527 1/20 0.44
FKBP4 Q02790 1/20 0.44
FKBP5 Q13451 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
CHRNA7 P36544 1/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 1/20 0.43
KMT2A Q03164 1/20 0.43
POLB P06746 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6160650 0.84 CYP2A6 (0.51) CYP2A6PTAFRHRH1CYP3A4CYP2D6
SCHEMBL6165461 0.82 ALDH1A1 (0.55) CYP2A6PTAFRHRH1CYP3A4CYP2D6
SCHEMBL6159742 0.82 PTAFR (0.49) CYP2A6PTAFRHRH1CYP3A4CYP2D6
SCHEMBL6158950 0.79 CYP2A6 (0.59) CYP2A6HRH1CYP3A4CYP2D6SLC6A2
SCHEMBL9190506 0.76 ALDH1A1 (0.55) PTAFRALDH1A1GAAKMT2APOLB
SCHEMBL6161202 0.75 HRH1 (0.59) CYP2A6PTAFRHRH1CYP3A4CYP2D6
SCHEMBL6160644 0.74 PTAFR (0.49) CYP2A6PTAFRHRH1KDM4E
SCHEMBL6160319 0.74 CYP2A6 (0.64) CYP2A6HRH1CYP3A4CYP2D6SLC6A2
SCHEMBL6158967 0.73 PTAFR (0.52) PTAFRALDH1A1GAAKMT2APOLB
SCHEMBL7751155 0.71 G6PD (0.50) ALDH1A1KMT2AHPGDHTTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129070-A4 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL MYERS SQUIBB CO (US) 2005-03-02 EP disclosed
EP-1129070-A1 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-09-05 EP disclosed
US-6228872-B1 PEPTIDE-PROLYL ISOMERASE AND ROTAMASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2001-05-08 US disclosed
WO-2000027811-A1 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-05-18 WO disclosed