SCHEMBL6158967

SCHEMBL6158967

COc1cc(CCCNCCCc2cccnc2)cc(OC)c1OC

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTAFR P25105 5/20 0.52
ALDH1A1 P00352 3/20 0.51
GAA P10253 2/20 0.51
KMT2A Q03164 1/20 0.51
KDM4E B2RXH2 1/20 0.48
POLB P06746 1/20 0.48
HPGD P15428 1/20 0.48
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
CHRM2 P08172 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
HSD17B10 Q99714 1/20 0.46
NOS1 P29475 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9190506 0.87 ALDH1A1 (0.55) PTAFRALDH1A1GAAKMT2AKDM4E
SCHEMBL6160639 0.85 PTAFR (0.59) PTAFRALDH1A1KDM4ECHRM2L3MBTL1
SCHEMBL16606319 0.81 CHRM2 (0.68) CHRM2TDP1L3MBTL1NOS1
SCHEMBL6159739 0.80 CHRM2 (0.56) PTAFRKMT2ACHRM2TDP1
SCHEMBL6165459 0.80 KMT2A (0.54) PTAFRALDH1A1GAAKMT2APOLB
SCHEMBL6158945 0.77 SIGMAR1 (0.68) CHRM2TDP1L3MBTL1
SCHEMBL6160313 0.74 SIGMAR1 (0.68) PTAFRCHRM2TDP1L3MBTL1
SCHEMBL6157737 0.74 SIGMAR1 (0.70) CHRM2TDP1L3MBTL1
SCHEMBL10730509 0.74 CYP2A6 (0.74) CHRM2TDP1L3MBTL1NOS1
SCHEMBL6161198 0.74 SIGMAR1 (0.68) PTAFRCHRM2TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129070-A4 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL MYERS SQUIBB CO (US) 2005-03-02 EP disclosed
EP-1129070-A1 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-09-05 EP disclosed
US-6228872-B1 PEPTIDE-PROLYL ISOMERASE AND ROTAMASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2001-05-08 US disclosed
WO-2000027811-A1 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-05-18 WO disclosed