SCHEMBL6159615

SCHEMBL6159615

c1ccc2c(c1)CN(c1ccnc3ccccc13)C2

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 2/20 0.61
ADRB2 P07550 1/20 0.61
KCNH2 Q12809 2/20 0.49
NUDT1 P36639 1/20 0.48
AR P10275 1/20 0.44
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HPGD P15428 1/20 0.43
EGFR P00533 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.42
PDGFRB P09619 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PKM P14618 1/20 0.41
ALOX15 P16050 1/20 0.41
CASP1 P29466 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6159074 0.98 NCF1 (0.59) NCF1ADRB2KCNH2NUDT1AR
SCHEMBL6159581 0.89 NUDT1 (0.63) NCF1ADRB2KCNH2NUDT1LMNA
Hydrochloric Acid SCHEMBL6162260 0.88 NUDT1 (0.61) NCF1ADRB2KCNH2NUDT1LMNA
SCHEMBL6160844 0.85 PKM (0.52) NCF1ADRB2KCNH2ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL6163063 0.84 PKM (0.51) NCF1ADRB2KCNH2ALDH1A1SMN1; SMN2
SCHEMBL3649189 0.80 NCF1 (0.73) NCF1ADRB2KCNH2ALDH1A1SMN1; SMN2
SCHEMBL14515644 0.80 NCF1 (0.73) NCF1ADRB2KCNH2ARALDH1A1
SCHEMBL6126024 0.80 NCF1 (0.51) NCF1ADRB2KCNH2NUDT1PDGFRB
SCHEMBL10268352 0.79 NCF1 (0.67) NCF1ADRB2KCNH2PDGFRBADRA2A
SCHEMBL19000048 0.79 NCF1 (0.71) NCF1ADRB2KCNH2ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1090917-B1 Quinolin-4-yl derivatives and their use as NMDA-receptor subtype blockers HOFFMANN LA ROCHE (CH) 2005-12-21 EP claimed
CN-1162424-C Quinoline-4-radical derivative II - 2004-08-18 CN claimed
US-6339093-B1 Isoquinoline derivatives HOFFMANN-LA ROCHE INC. 2002-01-15 US claimed
CN-1304936-A Quinoline-4-radical derivative II HOFFMANN LA BOCHE & CO AG F (CH) 2001-07-25 CN claimed
EP-1090917-A1 Quinolin-4-yl derivatives and their use as NMDA-receptor subtype blockers F. HOFFMANN-LA ROCHE AG (CH) 2001-04-11 EP claimed
EP-1090917-B1 Quinolin-4-yl derivatives and their use as NMDA-receptor subtype blockers HOFFMANN LA ROCHE (CH) 2005-12-21 EP disclosed
CN-1162424-C Quinoline-4-radical derivative II - 2004-08-18 CN disclosed
US-6339093-B1 Isoquinoline derivatives HOFFMANN-LA ROCHE INC. 2002-01-15 US disclosed
CN-1304936-A Quinoline-4-radical derivative II HOFFMANN LA BOCHE & CO AG F (CH) 2001-07-25 CN disclosed
EP-1090917-A1 Quinolin-4-yl derivatives and their use as NMDA-receptor subtype blockers F. HOFFMANN-LA ROCHE AG (CH) 2001-04-11 EP disclosed