SCHEMBL6160520

SCHEMBL6160520

COC(=O)[C@H](COCc1ccccc1)NCc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 4/20 0.49
TACR1 P25103 4/20 0.47
KCNT1 Q5JUK3 1/20 0.46
TRPM8 Q7Z2W7 1/20 0.45
ATM Q13315 2/20 0.44
PPARA Q07869 1/20 0.44
MAPK14 Q16539 1/20 0.43
LTA4H P09960 1/20 0.43
HPGD P15428 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6160524 1.00 S1PR1 (0.49) S1PR1TACR1KCNT1TRPM8ATM
SCHEMBL207075 0.91 TACR1 (0.54) TACR1TRPM8ATMALDH1A1HTT
SCHEMBL207074 0.91 TACR1 (0.54) TACR1TRPM8ATMALDH1A1HTT
SCHEMBL5055739 0.86 CA12 (0.55) TACR1TRPM8ATMPPARAL3MBTL1
SCHEMBL6160452 0.85 ATM (0.58) KCNT1TRPM8ATMPPARAL3MBTL1
SCHEMBL6160451 0.85 ATM (0.58) KCNT1TRPM8ATMPPARAL3MBTL1
SCHEMBL2717201 0.82 TACR1 (0.53) TACR1ATMPPARAALDH1A1HTT
SCHEMBL6158794 0.81 CTSK (0.47) KCNT1ATMMAPK14
SCHEMBL6158798 0.81 CTSK (0.47) KCNT1ATMMAPK14
SCHEMBL207546 0.80 TACR1 (0.47) TACR1ATMALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-20040157894-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-08-12 US disclosed
US-6699881-B2 MATRIX METALLOPROTEASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-03-02 US disclosed
US-20030078253-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2003-04-24 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-1132379-A1 NOVEL THIOL DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND UTILIZATION THEREOF Takeda Chemical Industries, Ltd. (JP) 2001-09-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078253-A1 Thiol compounds, their production and use TST, QSOX1, SULT1E1 S1PR1 2007/4885TACR1 782/4885KCNT1 535/4885
US-20040157894-A1 Thiol compounds, their production and use TST, SULT1E1, QSOX1 S1PR1 2052/4885TACR1 889/4885KCNT1 609/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.