SCHEMBL6160639

SCHEMBL6160639

COc1ccc(CCCCNCCCc2cccnc2)cc1OC

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTAFR P25105 11/20 0.59
MAPK1 P28482 1/20 0.55
SLC2A1 P11166 1/20 0.53
LMNA P02545 1/20 0.52
ALDH1A1 P00352 3/20 0.51
KDM4E B2RXH2 1/20 0.51
GLA P06280 1/20 0.51
NPSR1 Q6W5P4 2/20 0.50
HTT P42858 1/20 0.50
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
MAPT P10636 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CHRM2 P08172 1/20 0.49
USP2 O75604 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6158967 0.85 PTAFR (0.52) PTAFRLMNAALDH1A1KDM4ECHRM2
Hydrochloric Acid SCHEMBL9782076 0.81 SLC2A1 (0.65) SLC2A1ALDH1A1KDM4EGLACYP1A2
SCHEMBL6159739 0.81 CHRM2 (0.56) PTAFRCHRM2
SCHEMBL6165459 0.80 KMT2A (0.54) PTAFRALDH1A1CHRM2L3MBTL1
SCHEMBL11811971 0.79 SLC2A1 (0.68) SLC2A1ALDH1A1KDM4EGLACYP3A4
SCHEMBL16606319 0.79 CHRM2 (0.68) CYP1A2CYP3A4CYP2D6CHRM2L3MBTL1
SCHEMBL27432980 0.78 KDM4E (0.66) SLC2A1ALDH1A1KDM4EGLAMAPT
Hydrochloric Acid SCHEMBL7279779 0.78 SLC2A1 (0.83) SLC2A1
SCHEMBL6160313 0.78 SIGMAR1 (0.68) PTAFRCHRM2L3MBTL1
SCHEMBL6161198 0.78 SIGMAR1 (0.68) PTAFRCHRM2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129070-A4 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL MYERS SQUIBB CO (US) 2005-03-02 EP disclosed
EP-1129070-A1 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-09-05 EP disclosed
US-6228872-B1 PEPTIDE-PROLYL ISOMERASE AND ROTAMASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2001-05-08 US disclosed
WO-2000027811-A1 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-05-18 WO disclosed