SCHEMBL6160954

SCHEMBL6160954

COC(=O)[C@H](Cc1ccc(-c2nccs2)cc1)NC(=O)C(CSC(=O)c1ccccc1)CC(C)C

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BIRC2 Q13490 1/20 0.43
MMP9 P14780 3/20 0.42
MMP8 P22894 3/20 0.42
MMP2 P08253 3/20 0.42
ALDH1A1 P00352 1/20 0.42
THRB P10828 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TSHR P16473 1/20 0.40
MMP1 P03956 1/20 0.40
MME P08473 1/20 0.40
ACE P12821 1/20 0.40
CPA1 P15085 1/20 0.40
ACE2 Q9BYF1 1/20 0.40
MMP3 P08254 1/20 0.40
MMP7 P09237 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6160534 0.92 ALDH1A1 (0.44) BIRC2ALDH1A1THRBCYP2C9CYP2C19
SCHEMBL6161299 0.92 ALDH1A1 (0.44) BIRC2ALDH1A1THRBCYP2C9CYP2C19
SCHEMBL6160013 0.92 ALDH1A1 (0.44) BIRC2ALDH1A1THRBCYP2C9CYP2C19
SCHEMBL6160532 0.89 HDAC1 (0.39) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL6160530 0.89 HDAC1 (0.39) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL6165686 0.87 HDAC1 (0.38) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL6162653 0.87 MMP12 (0.43) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL6165693 0.87 HDAC1 (0.38) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL6162656 0.87 MMP12 (0.43) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL6165484 0.85 NPC1 (0.39) ALDH1A1THRBCYP2C9CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5994539-A Mercapto acyl aminoacid derivatives endowed with dual ACE-NEP inhibitory activity, useful in the treatment of cardiovascular diseases ZAMBON GROUP S.P.A. (IT) 1999-11-30 US claimed
EP-0877740-B1 THIOL DERIVATIVES WITH METALLOPEPTIDASE INHIBITORY ACTIVITY ZAMBON SPA (IT) 2005-03-30 EP disclosed
US-5994539-A Mercapto acyl aminoacid derivatives endowed with dual ACE-NEP inhibitory activity, useful in the treatment of cardiovascular diseases ZAMBON GROUP S.P.A. (IT) 1999-11-30 US disclosed