SCHEMBL6165484

SCHEMBL6165484

COC(=O)C(Cc1ccc(-c2nccs2)cc1)NC(=O)C(CSC(=O)c1ccccc1)Cc1cc(C)no1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
HDAC1 Q13547 4/20 0.37
HDAC6 Q9UBN7 4/20 0.37
ALDH1A1 P00352 2/20 0.36
ERAP2 Q6P179 1/20 0.36
ERAP1 Q9NZ08 1/20 0.36
LNPEP Q9UIQ6 1/20 0.36
LMNA P02545 1/20 0.36
GLA P06280 1/20 0.36
GABRA5 P31644 1/20 0.36
ACE P12821 4/20 0.36
ECE1 P42892 4/20 0.36
MME P08473 3/20 0.36
MMP13 P45452 3/20 0.36
THRB P10828 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6165492 1.00 NPC1 (0.39) NPC1RAB9AHDAC1HDAC6ALDH1A1
SCHEMBL6160534 0.89 ALDH1A1 (0.44) RAB9AALDH1A1LMNAGLAMME
SCHEMBL6160013 0.89 ALDH1A1 (0.44) RAB9AALDH1A1LMNAGLAMME
SCHEMBL6161299 0.89 ALDH1A1 (0.44) RAB9AALDH1A1LMNAGLAMME
SCHEMBL6165693 0.87 HDAC1 (0.38) HDAC1HDAC6ALDH1A1THRBCYP2C9
SCHEMBL6165686 0.87 HDAC1 (0.38) HDAC1HDAC6ALDH1A1THRBCYP2C9
SCHEMBL6160532 0.87 HDAC1 (0.39) HDAC1HDAC6ALDH1A1THRBCYP2C9
SCHEMBL6160530 0.87 HDAC1 (0.39) HDAC1HDAC6ALDH1A1THRBCYP2C9
SCHEMBL6160954 0.85 BIRC2 (0.43) ALDH1A1ACEMMETHRBCYP2C9
SCHEMBL6162656 0.84 MMP12 (0.43) ALDH1A1MMETHRBCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0877740-B1 THIOL DERIVATIVES WITH METALLOPEPTIDASE INHIBITORY ACTIVITY ZAMBON SPA (IT) 2005-03-30 EP disclosed