SCHEMBL6162045

SCHEMBL6162045

CC(C)(C)[Si](C)(C)OC1CCC(=O)N(Cc2ccc(Oc3ccccc3)cc2)C1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.44
HCRTR2 O43614 4/20 0.44
FAAH O00519 1/20 0.39
MGLL Q99685 1/20 0.39
THRB P10828 1/20 0.39
GRM2 Q14416 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CNR2 P34972 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GFER P55789 1/20 0.36
LTA4H P09960 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17061906 0.88 GRM2 (0.45) HCRTR1HCRTR2THRBGRM2L3MBTL1
SCHEMBL16759335 0.88 GRM2 (0.45) HCRTR1HCRTR2THRBGRM2L3MBTL1
SCHEMBL9061278 0.79 TSHR (0.50) THRBNPC1RAB9AALDH1A1
SCHEMBL31172328 0.79 TSHR (0.50) THRBNPC1RAB9AALDH1A1
SCHEMBL6162323 0.79 HCRTR1 (0.47) HCRTR1HCRTR2GRM2L3MBTL1EGLN1
SCHEMBL6159369 0.76 HCRTR1 (0.49) HCRTR1HCRTR2FAAHNPC1RAB9A
SCHEMBL6158683 0.76 HCRTR1 (0.49) HCRTR1HCRTR2FAAHGRM2NPC1
SCHEMBL28666165 0.73 HPGD (0.40) THRBGRM2RAB9AL3MBTL1
SCHEMBL28666162 0.73 HPGD (0.40) THRBGRM2RAB9AL3MBTL1
SCHEMBL17062216 0.73 P2RX7 (0.43) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-20040157894-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-08-12 US disclosed
US-6699881-B2 MATRIX METALLOPROTEASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-03-02 US disclosed
US-20030078253-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2003-04-24 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-1132379-A1 NOVEL THIOL DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND UTILIZATION THEREOF Takeda Chemical Industries, Ltd. (JP) 2001-09-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078253-A1 Thiol compounds, their production and use TST, QSOX1, SULT1E1 HCRTR1 1949/4885HCRTR2 1842/4885FAAH 3868/4885
US-20040157894-A1 Thiol compounds, their production and use TST, SULT1E1, QSOX1 HCRTR1 1930/4885HCRTR2 1754/4885FAAH 4084/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.