SCHEMBL6164260

SCHEMBL6164260

CC(Cc1nn(-c2ccccn2)c2c1C(=O)CC(C(C)C)C2)CC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CCNA2 P20248 8/20 0.38
CDK2 P24941 8/20 0.38
CCNO P22674 1/20 0.34
CCNE1 P24864 1/20 0.34
CCNA1 P78396 1/20 0.34
DHODH Q02127 1/20 0.33
CNR1 P21554 3/20 0.32
CNR2 P34972 3/20 0.32
BUB1 O43683 1/20 0.30
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
TP53 P04637 1/20 0.30
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6166197 0.89 CCNA2 (0.41) ALDH1A1SMN1; SMN2MAPTTHRBTDP1
SCHEMBL6168301 0.88 SMN1; SMN2 (0.43) ALDH1A1SMN1; SMN2MAPTTHRBTDP1
SCHEMBL6167945 0.86 DHODH (0.37) ALDH1A1SMN1; SMN2DHODHBUB1HPGD
SCHEMBL6164396 0.83 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2MAPTTHRBTDP1
SCHEMBL6163105 0.83 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2MAPTTHRBTDP1
SCHEMBL6164779 0.83 SMN1; SMN2 (0.44) ALDH1A1SMN1; SMN2MAPTTHRBTDP1
SCHEMBL6163771 0.82 CCNA2 (0.35) SMN1; SMN2CCNA2CDK2DHODHRAB9A
SCHEMBL6166206 0.82 OPRM1 (0.42) ALDH1A1SMN1; SMN2MAPTTHRBTDP1
SCHEMBL6771327 0.80 DHODH (0.32) DHODH
SCHEMBL6770749 0.80 SRC (0.35) ALDH1A1SMN1; SMN2DHODHKDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed