SCHEMBL6165464

SCHEMBL6165464

CCc1cccc(CC)c1Nc1nc2ccc(CC(=O)Nc3ccc(C(C)CC(=O)O)cn3)cc2o1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.37
GALK1 P51570 3/20 0.37
ITGA4 P13612 5/20 0.36
ITGB1 P05556 4/20 0.36
RIOK2 Q9BVS4 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CSNK1D P48730 1/20 0.35
IL6 P05231 1/20 0.35
STAT3 P40763 1/20 0.35
DEGS1 O15121 1/20 0.34
MAPT P10636 1/20 0.34
FFAR1 O14842 1/20 0.34
SOAT1 P35610 1/20 0.34
PDE4A P27815 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6167218 0.91 ITGA4 (0.41) HSD17B10GALK1ITGA4ITGB1MEN1
SCHEMBL6168715 0.91 LMNA (0.34) GALK1ITGA4LMNAPOLBIL6
SCHEMBL6165328 0.89 HSD17B10 (0.41) HSD17B10GALK1ITGA4ITGB1MEN1
SCHEMBL6164091 0.89 HSD17B10 (0.41) HSD17B10GALK1ITGA4ITGB1MEN1
SCHEMBL6165451 0.86 KMT2A (0.42) HSD17B10GALK1ITGA4ITGB1RIOK2
SCHEMBL6161852 0.86 ITGA4 (0.42) GALK1ITGA4ITGB1MEN1KMT2A
SCHEMBL6164820 0.86 ITGA4 (0.47) GALK1ITGA4ITGB1LMNAPOLB
SCHEMBL6170579 0.85 ITGB3 (0.39) HSD17B10GALK1ITGA4ITGB1POLB
SCHEMBL6165024 0.85 GALK1 (0.44) GALK1ITGA4ITGB1CSNK1DMAPT
SCHEMBL6165027 0.85 GALK1 (0.44) GALK1ITGA4ITGB1CSNK1DMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183254-B1 SUBSTITUTED BICYCLIC HETEROARYL COMPOUNDS AS INTEGRIN ANTAGONISTS AVENTIS PHARMA LTD (GB) 2005-01-12 EP disclosed
EP-1183254-A1 SUBSTITUTED BICYCLIC HETEROARYL COMPOUNDS AS INTEGRIN ANTAGONISTS Aventis Pharma Limited (GB) 2002-03-06 EP disclosed
WO-2000061580-A1 SUBSTITUTED BICYCLIC HETEROARYL COMPOUNDS AS INTEGRIN ANTAGONISTS AVENTIS PHARMA LIMITED (GB) 2000-10-19 WO disclosed