SCHEMBL6165500

SCHEMBL6165500

CC1(C)CCC(=O)c2c(-c3ccccc3)nn(CC(F)(F)F)c21

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.38
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
POLQ O75417 2/20 0.34
BUB1 O43683 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
SRC P12931 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ALOX15 P16050 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP19A1 P11511 2/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA1 P30542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6167609 0.90 CDC7 (0.37) BUB1ALDH1A1
SCHEMBL6166169 0.87 METAP2 (0.34) PTGS2POLQ
SCHEMBL6165166 0.85 USP19 (0.33) PTGS2KMT2APOLQALDH1A1
SCHEMBL6167324 0.85 BRD4 (0.38) MEN1KMT2ASRCTSHRHSD17B10
SCHEMBL6163427 0.82 POLL (0.34) POLQALDH1A1
SCHEMBL6161815 0.82 ADORA1 (0.38) MEN1KMT2ASMN1; SMN2TSHRHSD17B10
SCHEMBL6164754 0.82 EEF2K (0.34) MEN1KMT2APOLQHSD17B10ALOX15
SCHEMBL6163503 0.81 PTGS2 (0.40) PTGS2MEN1KMT2ASMN1; SMN2POLQ
SCHEMBL6165739 0.81 AURKA (0.31)
SCHEMBL6164080 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed