SCHEMBL6165525

SCHEMBL6165525

Cc1nn(CCO)c2c1C(=O)CC(C)(C)C2

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.61
HDAC1 Q13547 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
OPRM1 P35372 17/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 1/20 0.49
OPRK1 P41145 2/20 0.44
OPRD1 P41143 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6164718 0.82 HTT (0.41) HTTHDAC1HDAC6OPRM1KMT2A
SCHEMBL6164113 0.82 OPRM1 (0.49) HTTHDAC1HDAC6OPRM1KMT2A
SCHEMBL6164100 0.82 HDAC1 (0.45) HTTHDAC1HDAC6OPRM1KMT2A
SCHEMBL6162828 0.81 ALPL (0.63) HTTHDAC1HDAC6OPRM1KMT2A
SCHEMBL6166123 0.80 ALPL (0.43) HTTHDAC1HDAC6OPRM1KMT2A
SCHEMBL6166168 0.78 OPRM1 (0.55) HTTHDAC1HDAC6OPRM1KMT2A
SCHEMBL6165167 0.76 HTT (1.00) HTTHDAC1HDAC6OPRM1
SCHEMBL6163085 0.75 HDAC1 (0.68) HTTHDAC1HDAC6OPRM1KMT2A
SCHEMBL6165665 0.74 ALPL (0.39) HTTHDAC1HDAC6OPRM1KMT2A
SCHEMBL6166699 0.73 HTT (0.61) HTTHDAC1HDAC6OPRM1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed