SCHEMBL6166769

SCHEMBL6166769

Nc1[c]ccc(-c2cccnc2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 4/20 0.58
MKNK2 Q9HBH9 4/20 0.58
MEN1 O00255 1/20 0.58
PSIP1 O75475 1/20 0.58
AXL P30530 1/20 0.58
CYP2A6 P11509 5/20 0.54
CYP3A4 P08684 3/20 0.54
ALDH1A1 P00352 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP11B1 P15538 5/20 0.47
CYP11B2 P19099 5/20 0.47
CYP19A1 P11511 2/20 0.47
CYP17A1 P05093 1/20 0.47
PIK3CD O00329 1/20 0.45
PIP5K1C O60331 1/20 0.45
PIK3CA P42336 1/20 0.45
PI4KA P42356 1/20 0.45
PI4KB Q9UBF8 1/20 0.45
CYP2C9 P11712 2/20 0.44
CYP2B6 P20813 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27008286 0.79 CYP2A6 (0.54) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL23166247 0.79 CYP2A6 (0.54) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL27810982 0.79 CYP2A6 (0.54) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL9958246 0.77 CYP2A6 (0.52) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL6169243 0.77 LMNA (0.46) MEN1CYP3A4ALDH1A1CYP1A2CYP11B1
SCHEMBL3296186 0.77 MAOA (0.48) MEN1CYP3A4ALDH1A1PIK3CAPI4KA
SCHEMBL8125222 0.76 CYP11B2 (0.54) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL9957721 0.74 CYP2A6 (0.58) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL17951830 0.74 CYP2A6 (0.79) MKNK1MKNK2MEN1PSIP1AXL
SCHEMBL30620885 0.74 CYP2A6 (0.79) MKNK1MKNK2MEN1PSIP1AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542975-A2 9-CYANO-SUBSTITUTED PERYLENE-3,4-DICARBOXYLIC ACID MONOIMIDES BASF AKTIENGESELLSCHAFT (DE) 2005-06-22 EP disclosed
EP-1532210-A1 RYLENE DYES BASF AKTIENGESELLSCHAFT (DE) 2005-05-25 EP disclosed
EP-1513841-A1 1,6,9,14-TETRASUBSTITUTED TERRYLENE TETRACARBOXYLIC ACID DIIMIDES BASF AKTIENGESELLSCHAFT (DE) 2005-03-16 EP disclosed
WO-2004029028-A2 9-CYANO-SUBSTITUTED PERYLENE-3,4-DICARBOXYLIC ACID MONOIMIDES AS DYESTUFFS BASF AKTIENGESELLSCHAFT (DE) 2004-04-08 WO disclosed
WO-2004026965-A1 RYLENE DYES BASF AKTIENGESELLSCHAFT (DE) 2004-04-01 WO disclosed
EP-1373214-A1 RYLENE DERIVATIVES AND THEIR USE AS DYES BASF AKTIENGESELLSCHAFT (DE) 2004-01-02 EP disclosed
WO-2003104232-A1 1,6,9,14-TETRASUBSTITUTED TERRYLENE TETRACARBOXYLIC ACID DIIMIDES BASF AKTIENGESELLSCHAFT (DE) 2003-12-18 WO disclosed
EP-1370612-A2 THERMOCHROMIC RYLENE DYES BASF AKTIENGESELLSCHAFT (DE) 2003-12-17 EP disclosed
WO-2002068538-A2 THERMOCHROMIC RYLENE DYES BASF AKTIENGESELLSCHAFT (DE) 2002-09-06 WO disclosed
WO-2002066438-A1 RYLENE DERIVATIVES AND THEIR USE AS DYES BASF AKTIENGESELLSCHAFT (DE) 2002-08-29 WO disclosed
EP-1206456-A1 THERMOCHROMIC RYLENE DYES BASF AKTIENGESELLSCHAFT (DE) 2002-05-22 EP disclosed
WO-2001016109-A1 THERMOCHROMIC RYLENE DYES BASF AKTIENGESELLSCHAFT (DE) 2001-03-08 WO disclosed
EP-0804507-A1 SUBSTITUTED QUATERRYLENE TETRACARBOXYLIC ACID DIIMIDES BASF AKTIENGESELLSCHAFT (DE) 1997-11-05 EP disclosed
WO-1996022332-A1 SUBSTITUTED QUATERRYLENE TETRACARBOXYLIC ACID DIIMIDES BASF AKTIENGESELLSCHAFT (DE) 1996-07-25 WO disclosed