SCHEMBL6169232

SCHEMBL6169232

CCOC(C)=NC(=O)c1cccc(F)c1.Cc1nc(-c2cccc(F)c2)n(-c2ccc(S(N)(=O)=O)cc2)n1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 4/20 0.45
CA9 Q16790 3/20 0.45
PTGS2 P35354 9/20 0.44
PTGS1 P23219 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA4 P22748 2/20 0.42
KDR P35968 1/20 0.41
CA7 P43166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6174360 0.90 CSNK1D (0.39) CHRNA7CA9PTGS2PTGS1CA1
SCHEMBL6161912 0.88 CA1 (0.49) CA9PTGS2PTGS1CA1CA2
SCHEMBL5203437 0.82 PTGS2 (0.60) PTGS2PTGS1CA1CA2CA4
SCHEMBL6171769 0.80 CHRNA7 (0.53) CHRNA7CA9PTGS2PTGS1CA1
SCHEMBL6172783 0.78 CHRNA7 (0.41) CHRNA7CA9PTGS2PTGS1CA1
SCHEMBL5206016 0.75 LMNA (0.52)
SCHEMBL5206138 0.75 LMNA (0.52)
SCHEMBL6172900 0.73 CA9 (0.47) CHRNA7CA9PTGS2CA1CA2
SCHEMBL5203693 0.71 PTGS2 (0.47) CHRNA7PTGS2PTGS1CA1CA2
SCHEMBL5203044 0.70 CA2 (0.61) CA9PTGS2CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458706-A4 DIARYL 1,2,4-TRIAZOLE DERIVATIVES AS A HIGHLY SELECTIVE CYCLOOXYGENASE-2 INHIBITOR CJ CORP (KR) 2005-06-08 EP disclosed
EP-1458706-A1 DIARYL 1,2,4-TRIAZOLE DERIVATIVES AS A HIGHLY SELECTIVE CYCLOOXYGENASE-2 INHIBITOR CJ Corp. (KR) 2004-09-22 EP disclosed
WO-2003055875-A1 DIARYL 1,2,4-TRIAZOLE DERIVATIVES AS A HIGHLY SELECTIVE CYCLOOXYGENASE-2 INHIBITOR CJ CORP. (KR) 2003-07-10 WO disclosed