SCHEMBL6169271

SCHEMBL6169271

Cc1ccnc(C(=O)c2[nH]c3ccc(F)cc3c2C(C)C(=O)O)c1

nearest known ligand 0.66

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.66
PTGS1 P23219 7/20 0.66
KIF11 P52732 1/20 0.40
GABRA1 P14867 2/20 0.39
GABRG2 P18507 2/20 0.39
GABRB3 P28472 2/20 0.39
GABRA5 P31644 2/20 0.39
GABRA3 P34903 2/20 0.39
GABRA2 P47869 2/20 0.39
GABRA4 P48169 1/20 0.38
GABRA6 Q16445 1/20 0.38
JAK2 O60674 2/20 0.38
MAP2 P11137 1/20 0.37
IDO1 P14902 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6181624 0.92 PTGS2 (0.66) PTGS2PTGS1KIF11
SCHEMBL6170712 0.91 PTGS2 (0.53) PTGS2PTGS1GABRA1GABRG2GABRB3
SCHEMBL6172560 0.87 PTGS2 (0.50) PTGS2PTGS1
SCHEMBL6171485 0.87 PTGS2 (0.56) PTGS2PTGS1KIF11
SCHEMBL6174674 0.85 PTGS2 (0.68) PTGS2PTGS1
SCHEMBL6171838 0.85 PTGS2 (0.67) PTGS2PTGS1KIF11GABRA1GABRG2
SCHEMBL6168891 0.85 PTGS2 (0.67) PTGS2PTGS1GABRA1GABRG2GABRB3
SCHEMBL7202770 0.85 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL6173175 0.85 PTGS2 (0.69) PTGS2PTGS1MAP2
SCHEMBL6172104 0.84 PTGS2 (0.53) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1045833-B1 2,3-SUBSTITUTED INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER (US) 2005-11-02 EP claimed
US-6608070-B1 Useful for treatment of medical condition in which prostaglandins are implicated as pathogens NAKAO KAZUNARI (JP) 2003-08-19 US claimed
US-6608070-B1 Useful for treatment of medical condition in which prostaglandins are implicated as pathogens NAKAO KAZUNARI (JP) 2003-08-19 US disclosed